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2-(1-ethylpiperidin-4-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]acetamide
2-amino-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylpyridine-4-carboxamide
[(2S)-1-[6-(2-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]pyrrolidin-2-yl]methanol
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
[5-methyl-7-(quinoxalin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
1-[4-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
1-(dimethylamino)-2-{4-[(3-ethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propan-2-ol
4-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-5-methyl-1-(4-methylphenyl)piperazin-2-one
(1S,6R)-9-(1,5-dimethyl-1H-indole-2-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
1-ethyl-2-{[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
2-({4-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-6-methylquinolin-4-ol
N-(5-fluoro-2-methylphenyl)-2,7-diazaspiro[4.5]decane-2-carboxamide
2-ethyl-8-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}-2,8-diazaspiro[4.5]decan-3-one
2-(2H-1,3-benzodioxol-5-yloxy)-N-methyl-N-(quinolin-5-ylmethyl)propanamide
1-(2-methoxyethyl)-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]piperidin-2-one
4-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-yl)pyridine
2-{[1-(4-fluoro-3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-imidazole
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)(2-phenyl-1-{1-[3-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}ethyl)amine
N,3-dimethyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-propyl-1H-pyrazole-4-carboxamide
6-cyclopropyl-2-(4-{[2-(3-methoxyphenyl)azetidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
3-[4-(2,4-difluorophenyl)-1H-pyrazol-5-yl]-1-[(4-methoxyphenyl)methyl]piperidine
5-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[(5-methylfuran-2-yl)methyl]-1H,4H-pyrazolo[3,4-d]imidazole
3-cyclopropyl-N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-1H-pyrazole-5-carboxamide
2-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-1,3-thiazole-4-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-2-(phenylamino)pyrimidine-5-carboxamide
3-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidine-1-carbonyl]-1,2-dihydroquinoxalin-2-one
2-methyl-7-[1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-2,7-diazaspiro[4.4]nonane
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
8-[2-(1H-imidazol-4-yl)ethyl]-9-oxo-N-phenyl-2,8-diazaspiro[5.5]undecane-2-carboxamide
2-amino-4-(2-methoxypyrimidin-5-yl)-8-phenyl-5,6,7,8-tetrahydroquinoline-3-carbonitrile
N-[1-(3-methylpyridin-2-yl)propan-2-yl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(dimethyl-1,2-oxazol-4-yl)acetamide
9-[(4-acetylphenyl)methyl]-2-benzyl-2,9-diazaspiro[5.5]undecan-3-one
2-(2-methoxyphenyl)-N-[3-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]pyrrolidine-1-carboxamide
N-({4-[2-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]phenyl}methyl)methanesulfonamide
2,3,5,6-tetramethyl-N-[1-(pyrazin-2-yl)propan-2-yl]benzamide
9-(cyclopropylmethyl)-1-methyl-4-(1H-pyrrole-2-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-methyl-1-(1-methyl-5-phenyl-1H-pyrazole-3-carbonyl)-4-(2-methylphenyl)piperazine
N-[3-(furan-2-yl)phenyl]-1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperidine-4-carboxamide
2-(4-{[2-(4-chlorophenyl)morpholin-4-yl]methyl}phenoxy)ethan-1-ol
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-[1,3-dioxo-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-methylpiperidine-3-carboxamide
methyl (2S,4R)-1-{[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)carbamoyl]methyl}-4-hydroxypyrrolidine-2-carboxylate
4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxy-N-methyl-N-(oxan-2-ylmethyl)benzamide
1-[5-({[(2-fluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(piperidin-1-yl)propan-2-ol
1-{5-[(2,3-dihydro-1H-inden-2-yl)amino]-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-2-yl}piperidin-4-ol
4-[3-(2-cyclopropyl-1H-imidazol-1-yl)phenyl]-1,3-thiazole
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-4-[(2-methoxyethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-[4-(3-ethoxy-5-fluorophenyl)phenyl]-N,N-dimethylacetamide
1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
9-methoxy-4-[(2-methoxypyrimidin-5-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine