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1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4-(pyridin-4-ylmethyl)-1,4-diazepane
1-[3-(3-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-hydroxyethan-1-one
3-(quinolin-8-yl)-4H-chromen-4-one
N-[(3S,4R)-1-[2-(3-methoxyphenoxy)acetyl]-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
1-{2-[(6-methyl-2-phenylpyrimidin-4-yl)amino]ethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
(3aR,6aR)-2-cyclopentyl-5-[(4-hydroxy-3-methylphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{4-[(2,4-dimethoxy-3-methylphenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
(2S,4S)-N-ethyl-1-(1H-imidazol-4-ylmethyl)-4-(5-methylthiophene-2-amido)pyrrolidine-2-carboxamide
methyl 4-({[(3S,5S)-1-benzyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]amino}methyl)benzoate
4-[3-(4-fluorophenoxy)azetidine-1-carbonyl]-1-(propan-2-yl)pyrrolidin-2-one
N-(2H-1,3-benzodioxol-5-yl)-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
4-[2-(azocan-1-yl)acetyl]-1-(4-methoxyphenyl)piperazin-2-one
1-({[(2-methylphenyl)methyl]carbamoyl}methyl)-1,4-diazepane-6-carboxylic acid
N-({1-[2-(2,4-dioxoimidazolidin-1-yl)acetyl]piperidin-3-yl}methyl)-4-fluorobenzamide
2-ethyl-8-(4-methanesulfonylbenzoyl)-2,8-diazaspiro[4.5]decan-3-one
{2-[6-(cyclopentylamino)pyridazin-3-yl]phenyl}methanol
N-{[4-methoxy-3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)-2-(thiophen-3-yl)acetamide
N-(1-{1-[1-(4-methylphenyl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenoxypropanamide
3-benzyl-5-[(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)methyl]-1H-1,2,4-triazole
(1S,5R)-6-(cyclobutylmethyl)-3-[3-(3-methoxyphenyl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-({[5-(1-benzofuran-2-yl)-1,2,4-triazin-3-yl]amino}methyl)-1-(2-methoxyethyl)pyrrolidin-2-one
3-(1-methylpiperidin-3-yl)-1-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazin-1-yl}propan-1-one
N-(1-hydroxybutan-2-yl)-2-[(2-methylprop-2-en-1-yl)oxy]-N-(pyridin-2-ylmethyl)benzamide
{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(oxolan-2-ylmethyl)propylamine
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N-methyl-2-(1-methyl-3-oxopiperazin-2-yl)acetamide
2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
3-[(2-fluorophenyl)formamido]-N-[1-(4-methoxyphenyl)propyl]-N-methylpropanamide
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1H-indole-3-carboxamide
3-(2-chlorophenoxy)-1-(4-methoxy-2-methylbenzoyl)azetidine
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
3-[1-(2H-1,3-benzodioxol-5-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-4-methyl-1,2,5-oxadiazole
N-({1-[(2-ethoxyphenyl)methyl]piperidin-3-yl}methyl)-2-(4-methoxyphenyl)acetamide
2-benzyl-8-[(3-hydroxypiperidin-3-yl)methyl]-2,8-diazaspiro[4.5]decan-1-one
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(2-methoxypyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(3,5-dimethylbenzoyl)-N-[1-(furan-2-yl)ethyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-{thieno[2,3-d]pyrimidin-4-yl}-decahydro-1,6-naphthyridin-2-one
N,N-dimethyl-5-[2-(thiophen-3-yl)acetyl]-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
ethyl 4-{[4-(thiophene-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazine-1-carboxylate
3-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-1-[4-(1,3-thiazol-4-yl)phenyl]urea
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}cyclopropan-1-amine
1-methyl-5-[(2-methylpropyl)amino]-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[4-(3,4-dichlorophenyl)piperazin-1-yl]-3-(pyridin-2-yl)propan-1-one
4-(2-methylphenoxy)-1-(1-methylpyrrolidine-3-carbonyl)piperidine-4-carboxylic acid
3-({[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)-N-methylpropanamide
N-[2-(2,4-difluorophenyl)-1-{1-[2-(2-methoxyphenoxy)acetyl]piperidin-4-yl}ethyl]-N-methylpropanamide
1-cyclohexyl-4-{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}piperazine
8-({1-[(4-fluorophenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)-1,3-dioxa-8-azaspiro[4.5]decan-2-one
1-ethyl-3-[2-(morpholin-4-yl)-2-oxoethyl]-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
2-{5-[6-(4-methyl-1H-pyrazol-1-yl)pyrimidin-4-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol