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N-ethyl-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]-N-(pyridin-4-ylmethyl)piperidin-3-amine
4,6-dimethyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
1-{3-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]phenyl}ethan-1-one
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-(oxolan-3-yl)propanamide
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
2-(2-methylpropyl)-8-{[3-(morpholin-4-yl)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
2-(6-methoxynaphthalen-2-yl)-4-[3-(1H-pyrazol-1-yl)propyl]morpholine
(3R,4R)-1-{3-[4-(3-chlorophenyl)piperazin-1-yl]propyl}-4-ethylpiperidine-3,4-diol
4-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-6-methylpyrimidin-2-amine
2-{2-[3-(2-methylphenyl)phenyl]-1H-imidazol-1-yl}ethan-1-ol
(1-{2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-3-yl)methanamine
1-[3-(morpholin-4-yl)propyl]-6-oxo-N-[(1-phenylcyclopentyl)methyl]piperidine-3-carboxamide
(3R,4S)-1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4-cyclopropylpyrrolidin-3-amine
1-(2-methoxyphenyl)-4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazin-2-one
N-[5-({[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]carbamoyl}amino)-2-methoxyphenyl]propanamide
4-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-{2,7-diazaspiro[4.5]decan-2-ylmethyl}-6,8-dimethyl-1,2-dihydroquinolin-2-one
(3S,4R)-1-{[1-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-3-methoxypiperidin-4-amine
1-benzyl-2-methyl-5-(2-methylpropanamido)-N-(2-methylpropyl)-1H-1,3-benzodiazole-7-carboxamide
N4-[3-(4-methoxyphenyl)propyl]-2-methylpyrimidine-4,6-diamine
1-(4-methoxyphenyl)-4-[3-(pyrimidin-4-yl)piperidin-1-yl]butane-1,4-dione
3-phenyl-N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]benzamide
N-methyl-1-phenyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]cyclopropane-1-carboxamide
2-(2-fluorophenoxymethyl)-N-[1-(pyridin-2-yl)propan-2-yl]-1,3-oxazole-4-carboxamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[3-(4-methylphenyl)benzoyl]pyrrolidin-3-yl]methanol
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-1-{3-methyl-3,9-diazaspiro[5.6]dodecan-9-yl}propan-1-one
3-methyl-N-[1-methyl-3-(pyridin-3-yl)-1H-pyrazol-5-yl]-2-oxo-1-oxa-3,7-diazaspiro[4.5]decane-7-carboxamide
2-[3-(trifluoromethyl)phenyl]-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}acetamide
(1S,5R)-3-(6-ethyl-2-methylquinoline-4-carbonyl)-3,9-diazabicyclo[3.3.2]decan-10-one
4-tert-butyl-N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)benzamide
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
8-(6-methylpyridine-3-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
4-[3-(methoxymethyl)pyrrolidine-1-carbonyl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole
2-(dimethylamino)-2-(4-fluorophenyl)-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]acetamide
6,8-dimethyl-3-{3-oxa-9-azaspiro[5.5]undecan-9-ylmethyl}-1,2-dihydroquinolin-2-one
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}naphthalene-2-carboxamide
7-{[4-(2-methylpropyl)phenyl]methyl}-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
3-phenyl-1-{5-propylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
{[5-(1-methanesulfonylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
3-{[1-(1-methoxypropan-2-yl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
5-[(4-benzylpiperidin-1-yl)methyl]-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-1,2-oxazole-3-carboxamide
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-(4-methanesulfonylphenyl)ethan-1-one
N-methyl-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
1-[cyclopropyl(4-methylpyridin-2-yl)methyl]-3-[1-methyl-3-(pyridin-3-yl)-1H-pyrazol-5-yl]urea
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N-methyl-5-(oxolan-2-yl)thiophene-2-carboxamide
N,2,8-trimethyl-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]quinoline-4-carboxamide
N-({8-[(3,5-dimethylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)acetamide
(3R,4R)-4-cyclobutyl-3-methyl-1-[(6-methylpyridin-2-yl)methyl]piperidin-4-ol
N-[(4-methoxyphenyl)methyl]-2-(morpholin-4-yl)-6-phenylpyridine-3-carboxamide