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8-(1-aminocyclopropanecarbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}(methyl)[(3-phenyl-1,2-oxazol-5-yl)methyl]amine
4-(2,2-diethylmorpholin-4-yl)-N-(2-methoxyethyl)pyridine-2-carboxamide
(3R,4S)-4-[ethyl(1H-indol-4-ylmethyl)amino]oxolan-3-ol
N-{[5-fluoro-7-(4-fluoro-3-methylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(methylsulfanyl)acetamide
2-(3-fluorophenoxymethyl)-N-methyl-N-(oxolan-2-ylmethyl)-1,3-oxazole-4-carboxamide
5-[1-(cyclohex-3-en-1-ylmethyl)-4-hydroxypiperidin-4-yl]-N-(3,4-dimethoxyphenyl)-1-benzofuran-2-carboxamide
4-(cyclopropylmethyl)-1-({2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidin-5-yl}methyl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-oxo-1,2-dihydroquinoline-4-carboxamide
7-[3-(phenylsulfanyl)propyl]-2-oxa-7-azaspiro[4.5]decan-8-one
5-chloro-6-[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]pyridine-3-carboxylic acid
methyl 1-[(3S,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-{[1-(3-methylbutyl)-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,3-benzothiazole
5-[1-(3,4-difluorobenzoyl)piperidin-4-yl]-5-(3-phenylpropyl)imidazolidine-2,4-dione
4-({4-methyl-5-[1-(piperidin-4-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
5-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-4-yl}-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
ethyl 6-[8-(cyclopropylmethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-2-carboxylate
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-methyloxolane-2-carboxamide
N-{4-[(methylcarbamoyl)methyl]phenyl}-4-phenylazepane-1-carboxamide
3-[(3S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-1-(thiomorpholin-4-yl)propan-1-one
2-methyl-1-{1-[4-(1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}-5-(trifluoromethyl)-1H-1,3-benzodiazole
2-(2H-1,2,3-benzotriazol-2-yl)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-(methylamino)-N-[3-(2-phenylacetamido)phenyl]acetamide
ethyl 4-{[3-(trifluoromethyl)phenyl]methyl}-1-[(2,3,4-trimethoxyphenyl)methyl]piperidine-4-carboxylate
3-{1-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}phenol
N-methyl-N-(oxan-4-ylmethyl)-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
6-(5-fluoro-2-methoxyphenyl)-N2-(4-methylphenyl)-1,3,5-triazine-2,4-diamine
5-(2-cyclopentylacetamido)-N,1-dimethyl-2-(oxolan-2-yl)-N-(thiophen-2-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
N-(2-hydroxybutyl)-1-(4,6,7-trimethylquinazolin-2-yl)piperidine-4-carboxamide
6-methyl-2-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}quinolin-4-ol
1'-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
3-{[2-(1-benzofuran-2-yl)-1H-imidazol-1-yl]methyl}-5-cyclopropyl-1,2-oxazole
2-methoxy-N-{[7-({4-[methyl(phenyl)amino]phenyl}methyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzamide
N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
5-tert-butyl-3-{[4-(thiophen-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-pyrazole
4-ethyl-3-{1-[(1R,4S)-1,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]heptane-4-carbonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}[(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
3-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[(3S)-2-oxoazepan-3-yl]benzamide
N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
N-(1-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methylthiophene-3-carboxamide
1-(5-chloropyridin-2-yl)-4-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)piperazine
N-(2-ethoxybutyl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
1-[3-(2-fluorophenyl)benzoyl]-4-[(3-methoxyphenyl)methyl]-1,4-diazepan-5-one
N-({8-[4-(2-methylpropyl)benzoyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)cyclohexanecarboxamide
5-methyl-1-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-5-phenylpiperidin-2-one
methyl 3-(furan-2-amido)-1-(3-methylbutyl)-5-{[1-(propan-2-yl)piperidin-4-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N2-[(4-tert-butyl-1,3-thiazol-2-yl)methyl]-N4-methylpyrimidine-2,4-diamine
5-(3-{4-azatricyclo[4.3.1.13,8]undecan-4-yl}-3-oxopropyl)-5-(naphthalen-1-ylmethyl)pyrrolidin-2-one
N-(3-chloro-2-methylphenyl)-2-{2-[(dimethylamino)methyl]-4-(pyrazin-2-yl)phenoxy}acetamide
2-(4-{[ethyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)amino]methyl}phenoxy)ethan-1-ol