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1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5-(oxan-4-yl)-4-phenyl-1H-imidazole
3-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidine-1-carbonyl}-4H-pyrido[1,2-a]pyrimidin-4-one
8-[(6-chloro-2H-chromen-3-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
(2S,4S)-4-amino-N,N-diethyl-1-[2-(pyridin-3-yl)acetyl]pyrrolidine-2-carboxamide
5-(3-acetylphenoxymethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
(3S,4S)-1-[(2H-1,3-benzodioxol-5-yl)carbamoyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
2-[({2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)methyl]-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
methyl (2S,3S)-2-[(5-{[(5-chloropyridin-3-yl)oxy]methyl}-1,2-oxazol-3-yl)formamido]-3-methylpentanoate
[(2S,6S)-4-[(2,6-dimethoxyphenyl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
2-chloro-4-({[2-(ethylsulfanyl)ethyl]carbamoyl}amino)benzamide
(1S,5R)-3-(1H-1,3-benzodiazol-2-ylmethyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-3-(3-methylphenyl)piperidine
N,1,4,6-tetramethyl-2-oxo-N-[1-(2-phenylethyl)piperidin-3-yl]-1,2-dihydropyridine-3-carboxamide
4-{[3-(2-hydroxyethyl)-4-(3-methylbutyl)piperazin-1-yl]methyl}-2,6-dimethoxyphenol
1-[(3S,4R)-4-methoxyoxolan-3-yl]-4-phenyl-5-[5-(1H-pyrazol-5-yl)furan-2-yl]-1H-imidazole
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
1-(2-methylpropyl)-8-(2-phenylethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{5-[1-(methoxymethyl)cyclopropyl]-1-(4-methoxyphenyl)-1H-1,2,4-triazol-3-yl}benzamide
2-[({5-[1-(furan-3-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
3,5-dimethyl-1-(2-{2-[2-(5-methylfuran-2-yl)phenyl]-1H-imidazol-1-yl}ethyl)-1H-1,2,4-triazole
2-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decan-6-one
2-{[6-(3-chlorophenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}-N-(propan-2-yl)acetamide
2-{4-[(dimethylamino)methyl]phenoxy}-4,6-dimethylpyridine-3-carbonitrile
(2S,4R)-4-amino-N,N-diethyl-1-(6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)pyrrolidine-2-carboxamide
[(2S,6S)-4-[(1-propyl-1H-imidazol-2-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
1-methyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(4-methylphenyl)-4-[2-(pyridin-2-yl)pyrimidine-5-carbonyl]piperazin-2-one
2-chloro-5-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}pyridine
1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
4'-[(4-methyl-1,3-thiazol-5-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}({[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl})amine
N-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-[(3-methoxyphenyl)methyl]piperidin-3-amine
N-[(3R,4S)-1-(2,3-dihydro-1H-indene-5-carbonyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
4,6-dimethyl-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
3-(3-methoxyphenyl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-pyrazole-4-carboxamide
1-[3-(hydroxymethyl)piperidin-1-yl]-3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propan-1-one
7-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-3-(thiophen-2-yl)propanamide
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
5-{1-[(3,4-dimethoxyphenyl)methyl]piperidin-4-yl}-5-ethyl-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
1-{5H,6H-benzo[h]quinazolin-2-yl}-N-ethyl-N-(2-hydroxyethyl)-5-methyl-1H-pyrazole-4-carboxamide
N-[2-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)quinolin-6-yl]acetamide
1-[(2-methoxy-5-{[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methyl}phenyl)methyl]-1H-1,2,4-triazole
6-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
3-{[(6-aminopyridin-3-yl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
1-[cyclohexyl(methyl)amino]-3-{3-[(4-methyl-1,4-diazepan-1-yl)methyl]phenoxy}propan-2-ol
(2S,4R)-4-amino-1-(2,3-dimethylquinoxaline-6-carbonyl)-N-ethylpyrrolidine-2-carboxamide
5-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-2-amine
N-[(2-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)-3-phenyl-1H-pyrazole-4-carboxamide