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1-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(thiophen-2-yl)propan-1-one
4-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole
2-benzyl-N-{1,9-dioxaspiro[5.5]undecan-4-yl}-1,3-thiazole-4-carboxamide
N-methyl-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyridin-2-amine
N-[(1S,2R)-2-(cycloheptylamino)cyclobutyl]-2-(2,5-dimethoxyphenyl)acetamide
3-(methanesulfonylmethyl)-1-(1,3-thiazol-2-ylmethyl)piperidine
1-(1H-pyrazole-4-carbonyl)-3-[3-(trifluoromethyl)benzoyl]piperidine
N-methyl-3-[2-(propan-2-yloxy)phenyl]benzamide
N,N-dimethyl-7-(3,4,5-trimethoxybenzoyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-cyclopropyl-2-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}acetamide
N6-cyclopentyl-N5-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N5-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-methyl-N-[4-(morpholin-4-yl)butyl]pyrimidin-2-amine
2-{4-[(4-ethoxyphenyl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
3-(1H-indol-3-yl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
6-{3-[(3,5-dimethoxyphenyl)methoxy]phenyl}-N-methylpyridine-2-carboxamide
(3S)-1-ethyl-4-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methylpiperazin-2-one
7-[(3,4-difluorophenyl)methyl]-2-(5-methyl-1,3-oxazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-fluoro-2-(morpholin-4-yl)quinolin-3-yl]methyl}-3,5-dimethoxybenzamide
(3S)-3-amino-3-{ethyl[2-(3-methylphenoxy)ethyl]carbamoyl}propanoic acid
2-{4-[(5-methylfuran-2-yl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
(1S,5R)-3-{[4-(2-aminoethyl)phenyl]methyl}-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(1S,6R)-3-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3,9-diazabicyclo[4.2.1]nonane
9-(2,1,3-benzoxadiazol-4-ylmethyl)-6-oxa-9-azaspiro[4.5]decane
N-[(6-chloropyridin-3-yl)methyl]-N-methyl-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
4-[(3-methoxyphenyl)methyl]-1-[(2E)-4-methylpent-2-en-1-yl]-1,4-diazepan-5-one
3-[1-methyl-5-(piperidin-1-yl)-1H-1,2,4-triazol-3-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(4-methylphenyl)methyl]acetamide
(2R)-2-amino-2-phenyl-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2-[4-(ethanesulfonyl)piperazin-1-yl]-4-(1-methyl-1H-pyrazol-4-yl)pyrimidine
4-methyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
1-(2-{1-[2-(4-chlorophenoxy)acetyl]piperidin-2-yl}ethyl)-N-cyclopropyl-1H-1,2,3-triazole-4-carboxamide
1-cyclopentyl-3-(3-fluorophenyl)-3-[2-oxo-2-(4-phenylpiperidin-1-yl)ethyl]pyrrolidine-2,5-dione
2-phenyl-N-[1-(pyridin-3-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-cyclopentyl-4-[2-(4-fluorophenoxy)ethyl]-1,4-diazepan-5-one
N-[2-(cyclohexylsulfanyl)ethyl]-3-(4,5-dimethyl-1H-pyrazol-3-yl)propanamide
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-propylpiperidine
2-oxo-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1-oxaspiro[4.4]nonane-4-carboxamide
1-{4-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]thiophen-2-yl}ethan-1-one
2-amino-4-[2-(dimethylamino)-1,3-thiazol-5-yl]-6-(2-fluorophenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-(4-acetylphenoxy)-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}acetamide
2-[(1S,5R)-6-[2-(4-fluorophenoxy)acetyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
3-{[1-(azepan-1-yl)-2-methylpropan-2-yl]carbamoyl}-5-methoxybenzoic acid
2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-1-(morpholin-4-yl)ethan-1-one
8-(1-benzothiophen-2-ylmethyl)-1-(3-methylbutyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-[(3,5-difluorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-3-ol
2,6-dimethyl-3-[4-(2-phenylethyl)piperidine-1-carbonyl]-1,4-dihydropyridin-4-one
8-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-{[5-(1-cyclopentylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}-4-methylpiperazine