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3-chloro-N-({1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl}methyl)pyridine-4-carboxamide
5-(2-chlorophenyl)-4-[1-(3-phenylpropyl)piperidin-3-yl]pyrimidine
1-(butan-2-yl)-N3-ethyl-N5-[(5-fluoro-2-methylphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-(4-{[3-(pyrrolidin-1-yl)piperidin-1-yl]methyl}phenyl)imidazolidin-2-one
N-[2-(benzyloxy)ethyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)-2-(1H-1,2,4-triazol-1-yl)acetamide
1-ethyl-5-(2-methoxyacetamido)-N-[3-(morpholin-4-yl)propyl]-2-(pyridin-3-yl)-1H-1,3-benzodiazole-7-carboxamide
1-(1-acetylpiperidin-4-yl)-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
N-[2-(4-methyl-1,3-thiazol-2-yl)ethyl]-2-(pyridin-4-yl)quinoline-4-carboxamide
N-[2-(1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)ethyl]acetamide
4-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-1,4-oxazepan-6-ol
methyl 2-[(5-cyclopropyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazol-4-yl)formamido]acetate
5-(4-benzoylpiperidine-1-carbonyl)-1-[2-(morpholin-4-yl)ethyl]piperidin-2-one
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-5-hydroxypyrazine-2-carboxamide
N-{[1-(dimethylamino)cyclohexyl]methyl}-1-ethyl-3-methyl-1H-pyrazole-5-carboxamide
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]benzamide
3-(2-chlorophenyl)-3-{2-[3-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-1-(3-methoxypropyl)pyrrolidine-2,5-dione
N-(2-{7-[(2-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2,4-dimethylbenzamide
3-[(3S,7S,8aS)-3-[(4-chlorophenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-fluoro-2-methylphenyl)urea
N-[(2,3-dimethylphenyl)methyl]-4-(4-methylphenoxy)piperidine-4-carboxamide
N-[1-(2-chlorophenyl)ethyl]-1-(2-methylpropyl)-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-amine
N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-4-methyl-1,2,5-oxadiazole-3-carboxamide
(3aS,6aS)-1-[2-(2-methylphenyl)benzoyl]-octahydropyrrolo[2,3-c]pyrrole
1-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-5-(oxolan-3-yl)-4-phenyl-1H-imidazole
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
(4aR,7aS)-4-[2-(4-hydroxyphenyl)acetyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
(1S,5R)-6-(cyclobutylmethyl)-3-[(2-methyl-1,3-thiazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
8-[2-(4-methyl-1H-pyrazol-1-yl)propanoyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-2-(dimethylamino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(4-chlorophenyl)-N-{[8-(3-methylbutanoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}cyclopropane-1-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propan-1-one
3-(oxolan-3-yl)-5-(1-phenyl-1H-1,2,3-triazol-4-yl)-1,2,4-oxadiazole
(2R,3S,6R)-5-{imidazo[1,2-a]pyridine-2-carbonyl}-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-benzyl-8-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-(2-oxoimidazolidin-1-yl)phenyl]-6-[3-(prop-2-en-1-yloxy)benzoyl]-6-azaspiro[2.5]octane-1-carboxamide
N-[(3-ethoxyphenyl)methyl]-N-ethyl-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-[(1-methyl-1H-imidazol-2-yl)(phenyl)methyl]acetamide
1-(2-{[(2,3,5-trimethyl-1H-indol-7-yl)methyl]amino}pyrimidin-4-yl)piperidin-4-ol
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[4-(morpholin-4-yl)butyl]acetamide
N-[3-(3-chlorophenyl)phenyl]-1-(cyclopropylmethyl)piperidine-4-carboxamide
2-[2-(2-fluorophenyl)benzoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(2,5-dimethoxyphenyl)acetamide
N-({1-[(2-methoxynaphthalen-1-yl)methyl]piperidin-3-yl}methyl)acetamide
(1s,4s)-4-(4-{3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1H-1,2,3-triazol-1-yl)cyclohexan-1-amine
6-{2-[(4-methylpiperazin-1-yl)methyl]phenoxy}pyridine-2-carbonitrile
3-(5-chloro-2-methoxypyridin-4-yl)-6-(4-fluorophenyl)pyridazine
3-(2-chlorophenyl)-1-cyclopentyl-3-{2-oxo-2-[4-(pyridin-4-yl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione