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N-methyl-3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
2-[(3-chlorophenyl)methyl]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]-1,3-benzoxazole-6-carboxamide
methyl 3-(2,3-dimethoxybenzoyl)-7-oxo-9-(pyridin-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(1S,5R)-6-(1,3-thiazol-4-ylmethyl)-3-[3-(thiophen-3-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-ethyl-N-(furan-3-ylmethyl)-N-methyl-5-[(pyridin-2-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[1-(2-methylpropyl)cyclopropyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
1-tert-butyl-N-[3-(3-methylphenyl)propyl]-5-oxopyrrolidine-3-carboxamide
3-ethoxy-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-4-(prop-2-en-1-yloxy)benzamide
(4R,6S)-4-methyl-6-(4-{1-[methyl(pyridin-3-ylmethyl)amino]-2-phenylethyl}piperidine-1-carbonyl)-1,3-diazinane-2-thione
1-(4-fluorophenyl)-4-[1-(3-phenylpropyl)piperidin-3-yl]piperazine
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-4-(1H-imidazol-1-yl)benzamide
1-{2-[3-(methylsulfanyl)phenyl]pyrimidin-4-yl}piperidin-3-ol
1-(2-chlorophenyl)-3-(1-{1-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
3-[2-(3-methoxyphenyl)ethyl]-1-(thiophene-3-carbonyl)piperidine
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)(methyl){[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}amine
3-{5-[2-(2-methoxyphenoxy)propan-2-yl]-1,2,4-oxadiazol-3-yl}-6-methylpyridazine
3-[(7-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]pyridine
1-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]-3-(morpholin-4-yl)propan-1-one
N-[(3R,4S)-4-cyclopropyl-1-(2-hydroxyethyl)pyrrolidin-3-yl]-1-(4-methoxyphenyl)cyclopropane-1-carboxamide
2,6-dimethoxy-N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
4-(2-methoxyethyl)-N-[2-(3-methylphenoxy)phenyl]piperazine-1-carboxamide
5-[3-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridin-2-amine
(2R,6S)-4-{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}-2,6-dimethylmorpholine
4-(4-{[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}piperidin-1-yl)-N-[2-(morpholin-4-yl)ethyl]benzamide
N-(2,2-difluoroethyl)-4-{[(3R,4R)-4-hydroxypyrrolidin-3-yl]sulfamoyl}benzamide
4-(1H-1,2,3-benzotriazole-5-carbonyl)-1-(3-chlorophenyl)-5-methylpiperazin-2-one
(1R,2S,6R,7S)-4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-azatricyclo[5.2.2.02,6]undecane
4,4-difluoro-N-(3-methanesulfonamido-4-methoxyphenyl)piperidine-1-carboxamide
1-{1-[2-(4-methoxyphenoxy)acetyl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-({7-[2-(4-methoxyphenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)propane-1-sulfonamide
N-[(2-aminopyrimidin-5-yl)methyl]-8-methoxy-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N,2-dimethyl-6-oxo-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-1,6-dihydropyrimidine-5-carboxamide
8-[5-(methoxymethyl)thiophene-2-carbonyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-[3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carboxamide
(2S)-2-amino-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)propanamide
3,3-dimethyl-1-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}butan-1-one
N,N-dimethyl-5-({4-[methyl(phenyl)amino]phenyl}methyl)-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N,N-dimethyl-3-{octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl}aniline
2-(5-chlorothiophene-2-carbonyl)-7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decane
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-methyl-N-[2-(oxan-2-yl)ethyl]propanamide
8-(2,4-difluorobenzoyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{5-[4-(1,3-benzoxazol-2-yl)piperazine-1-carbonyl]-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl}furan-2-carboxamide
N-cyclopentyl-3,4-difluoro-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}benzene-1-sulfonamide
1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-(1H-pyrrole-3-carbonyl)-1,4-diazepan-6-ol
N-[(3-fluorophenyl)methyl]-2-(3-methoxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-[1-(morpholine-2-carbonyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
1-methyl-4-(2-oxo-1-phenylpyrrolidine-3-carbonyl)piperazin-2-one
N-[3-(3,4-dimethoxyphenyl)propyl]-2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N,4-dimethyl-3-{[(3-phenylpropyl)(propan-2-yl)carbamoyl]amino}benzamide
N-[3-(5-methyl-4-{[(2,4,5-trifluorophenyl)formamido]methyl}-1,3-oxazol-2-yl)phenyl]pyridine-2-carboxamide