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dimethyl({[4-methyl-5-(1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl})amine
N-{1-[1-(1H-indol-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
7-(9H-fluoren-2-ylmethyl)-3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
4-[(1H-imidazol-2-ylmethyl)sulfamoyl]-N-(thiolan-3-yl)benzamide
N-[(2-methoxyphenyl)methyl]-1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{5-[2-(azocan-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-[4-(trifluoromethyl)phenyl]ethan-1-one
6-[(2-chloro-6-fluorophenyl)methyl]-N-(2-methoxyphenyl)-6-azaspiro[2.5]octane-1-carboxamide
3-hydroxy-2-methyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}benzamide
1-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
1-(4-methyl-2-{[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amino}pyrimidin-5-yl)ethan-1-one
8-(1H-imidazol-2-ylmethyl)-3-{3-[methyl(2-methylpropyl)amino]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-[1-(4-ethenylbenzoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
1-{2-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-oxoethyl}-5-methylpyrrolidin-2-one
N-[2-(dimethylamino)ethyl]-4-methoxy-3-{[1-(5-methylhex-5-en-2-yl)piperidin-4-yl]oxy}benzamide
N-[(2R,3R)-1'-(2,4-dimethylbenzoyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxybenzamide
({5-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-1,3,4-oxadiazol-2-yl}methyl)dimethylamine
2-(5-{[4-(3-methoxybenzoyl)piperazin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)pyrazine
1-{2-[1-(8-chloroquinolin-2-yl)piperidin-4-yl]ethyl}pyrrolidin-2-one
methyl 3-(2-fluorobenzoyl)-9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(furan-2-ylmethyl)pyrrolidin-3-yl]-2-methyl-1H-pyrrole-3-carboxamide
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-[(5-ethylfuran-2-yl)methyl]piperidine-4-carboxylic acid
1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-4-(hydroxymethyl)azepan-4-ol
4-(4-{[(2,2-dimethyl-1-phenylcyclopropyl)methyl]amino}piperidin-1-yl)-N-[2-(morpholin-4-yl)ethyl]benzamide
5,6-dimethoxy-2-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-1,2-dihydroisoquinolin-1-one
3-{3-[cyclohexyl(methyl)amino]propyl}-8-(oxan-3-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-methyl-1-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(1H-pyrazol-1-yl)propan-1-one
N-(6-methylpyridazin-3-yl)-4-{[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl}benzamide
2-{8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-N-(2-phenylethyl)acetamide
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(oxolan-3-yl)benzamide
1-{3-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-3-methoxypiperidine
1-(adamantan-1-yl)-4-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperazine
N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}pyridine-3-sulfonamide
methyl N-{2-[2-(4-fluorophenyl)piperidin-1-yl]-2-oxoethyl}carbamate
5-(2-methoxyacetamido)-N-[(3-methoxyphenyl)methyl]-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-methylpropanamide
N-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-[(3-methylpyridin-2-yl)methyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
(3-{2-[1-(2,6-difluorobenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
N-[(1R,3S)-3-(pyrrolidine-1-carbonyl)cyclopentyl]quinoline-4-carboxamide
N-{1-[1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxy-2-phenylacetamide
4-{4-[4-(dimethylamino)azepane-1-carbonyl]phenyl}-2-methylbutan-2-ol
7-fluoro-1-[2-(piperidin-1-yl)ethyl]-3-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
3-(3-amino-1H-indazol-1-yl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
9-(3-hydroxy-4-methylbenzoyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
[(2,6-difluoro-3-methylphenyl)methyl](ethyl)(oxan-4-ylmethyl)amine
2-(4-methylphenoxy)-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-3,4-dimethylbenzamide
5-(2-{[(4-fluorophenyl)methyl]amino}ethyl)-1-[2-(4-methoxyphenyl)ethyl]pyrrolidin-2-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-5-[3-(2-methylpropyl)-1,2-oxazol-5-yl]-1H-1,2,4-triazole