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N-(2-methoxyethyl)-1-[1-(6-methoxypyrimidin-4-yl)piperidin-4-yl]piperidine-3-carboxamide
1-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-cyclopropyl-3-[1-(1H-indol-3-ylmethyl)piperidin-3-yl]propanamide
2-(1-benzyl-3-oxopiperazin-2-yl)-N-(1-phenylpiperidin-4-yl)acetamide
methyl 5-[(5-chloro-2-hydroxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
1-(2-methoxyethyl)-3-(2-methylphenyl)-3-(2-oxo-2-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}ethyl)pyrrolidine-2,5-dione
4-[2-(1-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}piperidin-2-yl)ethyl]phenol
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-[2-(methylamino)ethyl]-1,2-oxazole-3-carboxamide
5-[1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-5-(3-phenylpropyl)imidazolidine-2,4-dione
methyl (2S)-1-{2-[4-(4-acetylphenyl)piperazin-1-yl]-6-(4-methylthiophen-2-yl)pyridine-3-carbonyl}pyrrolidine-2-carboxylate
3-methyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1-propyl-1H-pyrazole-4-carboxamide
N-(5-chloro-2-methoxyphenyl)-6,8-dioxo-2,7-diazaspiro[4.4]nonane-2-carboxamide
(4aR,7aS)-1-ethyl-4-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(furan-2-yl)-2-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamido]propanoic acid
methyl (2R,4S)-4-hydroxy-1-{[2-(2-phenylethynyl)phenyl]methyl}piperidine-2-carboxylate
2-cyclopropyl-4-hydroxy-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]pyrimidine-5-carboxamide
(4aS,8aS)-2-(3-fluoropyridin-4-yl)-decahydro-2,7-naphthyridin-4a-ol
3-[2-(2,2-diphenylethyl)morpholine-4-carbonyl]pyridin-2-ol
1-cyclopentyl-4-[(2-methoxynaphthalen-1-yl)methyl]piperazin-2-one
1-[(4-methanesulfonylphenyl)methyl]-3-(2-methylphenyl)pyrrolidin-3-ol
3-(dimethyl-1,2-oxazol-4-yl)-1-(7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
6-(propan-2-yl)-2-[3-(pyrrolidin-1-yl)piperidine-1-carbonyl]-1H-indole
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}propanamide
N-ethyl-2,6-dimethyl-N-(2-methylprop-2-en-1-yl)imidazo[1,2-a]pyridine-3-carboxamide
(1S,5R)-3-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(2R,3R)-2-methoxy-1'-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
1-(4-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)-2-phenoxyethan-1-one
N-[3-(1H-pyrazol-1-yl)propyl]-3-[(pyrrolidin-3-yl)sulfamoyl]benzamide
1-[2-(2,2-dimethyloxan-4-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-[2-(2-fluorophenyl)ethyl]piperidine-3-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-1-{2-[2-(3-{[methyl(quinolin-8-ylmethyl)amino]methyl}phenoxy)ethyl]piperidin-1-yl}ethan-1-one
3-(1H-1,2,3,4-tetrazol-1-yl)-N-[(1R,3S)-3-(thiomorpholine-4-carbonyl)cyclopentyl]propanamide
1-[1-(5-methylthiophene-2-carbonyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
N-cyclopropyl-N-[(4-hydroxyphenyl)methyl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N-ethyl-6-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-N-methylpyridine-3-carboxamide
3-[2-(dimethylamino)ethyl]-5-[1-(2,2-dimethylpropanoyl)piperidin-4-yl]-5-(3-methylbutyl)imidazolidine-2,4-dione
1-({4-[(3,5-difluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)-4-(pyridin-3-yl)piperidin-4-ol
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-(quinolin-4-ylformamido)acetic acid
1-{1-[3-(dimethylamino)pyrazin-2-yl]piperidin-4-yl}-3-methylbutan-1-ol
4-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-3-yl]benzoic acid
3-(azetidine-1-carbonyl)-N-methyl-N-[3-(oxolan-2-yl)propyl]benzene-1-sulfonamide
1-[2-(2-methyl-1,4-oxazepane-4-carbonyl)phenyl]ethan-1-one
2-(3-hydroxypropyl)-8-(6-methylquinolin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
5-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazine-1-carbonyl]-2-ethylpyrimidine
1-(1-benzyl-1H-pyrazole-4-carbonyl)-N-ethyl-N-(pyridin-4-ylmethyl)piperidin-3-amine
5-{1-[2-(4-methoxyphenyl)acetyl]piperidin-4-yl}-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
2-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-N-(2-methylbutan-2-yl)acetamide
(2E)-3-(1H-imidazol-4-yl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)prop-2-enamide
1,3-dimethyl-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-{[(4-{1-azabicyclo[3.2.1]octan-5-yloxy}phenyl)methyl]amino}-2-methylpropane-1,3-diol
N-methyl-2-[4-(pyridin-3-yl)-1H-pyrazol-1-yl]acetamide