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4-(2,3-dihydro-1,4-benzodioxin-6-yl)-5,6-dimethyl-2-(trifluoromethyl)pyrimidine
6-tert-butyl-N-({2-[(dimethylamino)methyl]phenyl}methyl)-N,1-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-6-phenyl-1,2-dihydropyridin-2-one
6,7-dimethoxy-3-({methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
N-[1-ethyl-7-(3-methoxypiperidine-1-carbonyl)-2-(pyridin-3-yl)-1H-1,3-benzodiazol-5-yl]-2-methoxyacetamide
9-[2-(1H-imidazol-1-yl)propanoyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(3S,4R)-4-(4-methylphenyl)-1-propanoylpyrrolidin-3-yl]acetamide
3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]propanamide
2-(1-{imidazo[1,2-a]pyridin-2-ylmethyl}-1H-imidazol-2-yl)-4-(propan-2-yl)-1,3-thiazole
1-{3-[(dimethylsulfamoyl)amino]phenyl}-3-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]urea
3-methyl-N-{1-[1-(5-methyl-1H-indole-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
N-[2-(2-chlorophenyl)ethyl]-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-methyl-N-[4-(morpholin-4-yl)butyl]acetamide
3-[2-({2-[(3-hydroxyphenyl)amino]-6-methylpyrimidin-4-yl}amino)ethyl]-1,3-oxazolidin-2-one
[(2-fluoro-4-methoxyphenyl)methyl](methyl)[3-(1-methyl-1H-imidazol-2-yl)propyl]amine
4-ethyl-3-{[1-(2-methyl-1H-1,3-benzodiazole-4-carbonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
(1R,3S)-7-(2,6-dimethylpyridine-4-carbonyl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
(1S,5R)-6-(1-methyl-1H-indole-3-carbonyl)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-[(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)methyl]-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
1-acetyl-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}piperidine-4-carboxamide
2-(3,5-difluorophenyl)-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylacetamide
5-methyl-3-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-indazole
N-({8-benzyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-3-phenyl-1,2-oxazole-5-carboxamide
5-{[2-(1-benzylpiperidin-4-yl)ethyl]carbamoyl}-1H-imidazole-4-carboxylic acid
N-[3-(1H-indazol-1-yl)propyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
N-[(5-chloro-2-methoxyphenyl)methyl]-N-ethyl-2-(ethylamino)pyrimidine-5-carboxamide
2-[2-(morpholin-4-yl)acetyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1-methyl-N-[2-(7-{[4-(methylsulfanyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]piperidine-3-carboxamide
1-{2-[methyl({7H-pyrrolo[2,3-d]pyrimidin-4-yl})amino]ethyl}piperidin-2-one
N-[(2-chlorophenyl)methyl]-1-(2-cyclohexylethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
(2E)-3-(3-fluorophenyl)-1-{3-[5-(2-fluorophenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}prop-2-en-1-one
1-(2-{[2-(dimethylamino)-2-(pyridin-2-yl)ethyl]amino}pyrimidin-4-yl)piperidin-4-ol
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-phenoxypropanamide
(1R,2S,4R)-N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
(1S,5R)-3-{2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]acetyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
2-phenyl-1-{4-[(3-phenyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}ethan-1-ol
1-{3,9-diazaspiro[5.5]undecan-3-yl}-2-[(2-methylphenyl)sulfanyl]ethan-1-one
(4aR,7aS)-1-methyl-4-[2-(1H-1,2,4-triazol-1-yl)benzoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
({1-benzyl-3-[(3,4-dimethoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)dimethylamine
9-(4-chloro-2-hydroxybenzoyl)-2-[2-(dimethylamino)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(cyclopent-2-en-1-yl)acetyl]-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
2-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-5-methylphenol
(2S)-1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-4-methyl-2-phenylpiperazine
2-(1-ethylpiperidin-4-yl)-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}acetamide
2-{4-[(2S)-2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]piperidin-1-yl}acetamide
5-(2-butylpyrrolidine-1-carbonyl)-4-ethyl-1,3-thiazol-2-amine
methyl 4-(methylsulfanyl)-2-{3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propanamido}butanoate
2-[3-(pyridin-4-yl)-5-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-yl)-1H-1,2,4-triazol-1-yl]acetic acid
5-(furan-2-yl)-1-(oxan-2-ylmethyl)-4-phenyl-1H-imidazole
4-{5-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyrimidin-2-yl}morpholine