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N-{4-[(2S)-2-amino-3-(1H-imidazol-4-yl)propanamido]phenyl}-4-methylbenzamide
[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)[(1-phenyl-1H-pyrazol-4-yl)methyl]amine
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)(ethyl)[2-(1H-pyrazol-1-yl)ethyl]amine
5-{1-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]pyrrolidin-2-yl}-N,N-dimethylthiophene-2-carboxamide
3-({5-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}methyl)pyridine
2-{4-[(2-chloro-4,5-dimethoxyphenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
5,6-dimethyl-N-[1-(pyridin-4-ylmethyl)piperidin-4-yl]pyrimidin-4-amine
4-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-methoxypyridine-3-carbonitrile
4-(4-{[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}phenyl)but-3-yn-1-ol
3-butyl-5-(5-ethoxyfuran-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-[1-(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2-methylbenzamide
5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-(3-phenylpropyl)-1,2-oxazole-3-carboxamide
N-[(4-hydroxyazepan-4-yl)methyl]-2-oxo-1,2-dihydroquinoline-3-carboxamide
1-benzyl-N,2-dimethyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-5-(2-methylpropanamido)-1H-1,3-benzodiazole-7-carboxamide
5-acetamido-N-(2-hydroxybutyl)-1-(2-methoxyethyl)-2-(pyridin-2-yl)-1H-1,3-benzodiazole-7-carboxamide
N-(1-benzofuran-2-ylmethyl)-1-[(2-fluorophenyl)methyl]piperidin-3-amine
4-(4-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-1-yl)butan-1-ol
2-(2-{1-[1-(pyridin-3-yl)propan-2-yl]-1H-imidazol-2-yl}phenoxy)acetic acid
({4-ethyl-5-[1-(5-methylpyrazine-2-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-ethyl-1,1-dioxo-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-1λ6-thiane-4-carboxamide
3-cyclopentyl-1-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}propan-1-one
4-{[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]methyl}benzoic acid
2-phenoxy-N-(1-{7-[(2,4,6-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
N-[(2-aminopyridin-3-yl)methyl]-3-(piperazine-1-carbonyl)benzene-1-sulfonamide
7-(oxolane-2-carbonyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-ethyl-5-{pyrazolo[1,5-a]pyridin-7-yl}thiophene-2-carboxamide
(3S,4R)-1-[(3-hydroxyphenyl)methyl]-4-phenylpyrrolidine-3-carboxylic acid
1-cyclopentyl-3-(3-fluorophenyl)-3-{2-oxo-2-[4-(propan-2-yl)piperazin-1-yl]ethyl}pyrrolidine-2,5-dione
N-[4-(1,3-thiazol-4-yl)phenyl]-1-[2-(4H-1,2,4-triazol-4-yl)ethyl]piperidine-3-carboxamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]acetamide
1-[3-(3-methylphenyl)piperidin-1-yl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
4-(1-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)thiomorpholine
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-(2-oxopyrrolidin-1-yl)butanamide
4-{[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]methyl}-3-methoxyphenol
{1-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]-2-phenylethyl}(2-methoxyethyl)(pyridin-3-ylmethyl)amine
3-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-1-tert-butyl-1H-pyrrole
6-methyl-2-[(2-methylphenyl)methyl]-3-(3-methylpiperidine-1-carbonyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridin-4-one
2-(2-methyl-1,3-thiazol-4-yl)-1-[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
(3aS,6aR)-5-(2,3-dihydro-1H-inden-2-yl)-3-[(2-methoxyphenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
ethyl 1-[2-(dimethylamino)ethyl]-5-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-methyl-1-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-5-one
2-[3-benzyl-1-(4-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-methyl-N-(propan-2-yl)acetamide
1-methyl-4-(1-{1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}ethyl)piperazine
3-ethyl-4-methyl-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-pyrazole-5-carboxamide
2-{4-[2-(dimethylamino)-2-(4-fluorophenyl)acetyl]piperazin-1-yl}benzonitrile
2-(4-carbamoylpiperidin-1-yl)-2-(2,6-dimethoxypyridin-3-yl)acetic acid
2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-3-carboxamide
N-[1-(pyrimidin-2-yl)piperidin-3-yl]-2-(pyrrolidin-1-yl)benzamide
3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(1-phenylcyclopentyl)methyl]propanamide
1-{3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidin-1-yl}-2-(pyrimidin-2-ylsulfanyl)ethan-1-one