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8-{2-[(4-methoxyphenyl)amino]-2-methylpropanoyl}-2,8-diazaspiro[4.5]decan-3-one
3-(4-methyl-1,3-thiazol-5-yl)-1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propan-1-one
(1S,5R)-N-cyclopentyl-7-oxo-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-{2-[2-(3-{[methyl(quinolin-8-ylmethyl)amino]methyl}phenoxy)ethyl]piperidin-1-yl}-2-(2-phenyl-1,3-thiazol-4-yl)ethan-1-one
(2S)-1-[2-(3-fluorophenyl)-1,3-benzoxazole-5-carbonyl]pyrrolidine-2-carboxamide
ethyl 1-[2-(2-methyl-1,3-thiazol-4-yl)acetamido]cyclobutane-1-carboxylate
N-{2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl}-2-(methylamino)pyrimidine-5-carboxamide
3-[(4-fluorophenyl)formamido]-N-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]propanamide
7-(5-chloropyridin-2-yl)-9-methoxy-4-(naphthalene-1-sulfonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-N,6-dimethylpyrimidin-2-amine
{[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)[(5-propyl-1H-pyrazol-3-yl)methyl]amine
2-amino-4-cyclopropyl-6-(pyridine-2-carbonyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]-2-(4-methyl-1,4-diazepan-1-yl)acetamide
N-(1,3-dimethyl-1H-pyrazol-5-yl)-4-(2-phenoxyethyl)piperazine-1-carboxamide
N,N-diethyl-2-{4-[2-(2-methoxyphenyl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}acetamide
(2R)-2-amino-N,4-dimethyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]pentanamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-methylquinoline-4-carboxamide
4'-methyl-1-(5-methylpyridine-3-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(2-methoxyphenyl)-2-methylpiperazine
methyl (2S,4R)-1-[(4-chlorophenyl)methyl]-4-(2-cyclopropylquinoline-4-amido)pyrrolidine-2-carboxylate
(adamantan-1-ylmethyl)({[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
N-[(5-chlorothiophen-2-yl)methyl]-5-[(3-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
(3R,9aR)-3-(2-methylpropyl)-8-(naphthalene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-{1-[2-(2,5-dimethoxyphenyl)acetyl]piperidin-4-yl}-5-ethyl-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
2-methyl-4-{5-[4-(4H-1,2,4-triazol-4-yl)piperidine-1-carbonyl]furan-2-yl}but-3-yn-2-ol
(3aR,7aS)-2-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-{2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}-3-(pyridin-4-yl)propan-1-one
2-{4-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]quinazolin-2-yl}ethan-1-amine
1-methyl-N-(piperidin-4-yl)-3-propyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
(2S)-5-oxo-N-{[7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pyrrolidine-2-carboxamide
2-[2-(butan-2-yl)phenoxy]-N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-N-methylacetamide
4-[(2S,4R)-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carbonyl]morpholine
3-(dimethoxy-1,3,5-triazin-2-yl)-5-methyl-1H-indole
1-(2-ethoxyethyl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
N-{4-[2-(2,5-dioxoimidazolidin-4-yl)acetamido]-2-methoxyphenyl}-3-methylbutanamide
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-2-(dimethylamino)-2-(4-fluorophenyl)-N-methylacetamide
5-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-benzylfuran-2-carboxamide
2-{[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]methyl}pyridine-3-carboxylic acid
N-({6-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]pyridin-3-yl}methyl)acetamide
2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]-4-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}morpholine
4-fluoro-2-methoxy-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}benzamide
1-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
N-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
N-(3,3-diphenylpropyl)-1-methyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-chloro-N-({8-cyclopropanecarbonyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-4-fluorobenzamide
[4-(3-phenylpropyl)-1-(quinolin-8-ylmethyl)piperidin-4-yl]methanol
1-(4-methylpyridine-3-carbonyl)-2-(pyrrolidine-1-carbonyl)piperazine
N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-4-methylpyrimidin-2-amine
1-[(2-fluorophenyl)methyl]-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
7-methoxy-3-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-1,2-dihydroquinolin-2-one