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4-(3-methylphenyl)-3-(1H-pyrazol-5-yl)-4H-1,2,4-triazole
1-benzyl-3-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}pyrrolidine
1-{[3-(3-methoxyphenyl)oxolan-3-yl]methyl}-4-(2-methylpyridin-4-yl)piperazine
2-{1-[(4-fluorophenyl)methyl]-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl}ethan-1-ol
methyl 2-(1,4-dioxan-2-ylmethyl)-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
2-{4-[({[(2R,3R,5S)-2-(4-chlorophenyl)-1-ethyl-5-(hydroxymethyl)-5-methylpyrrolidin-3-yl]methyl}amino)methyl]phenoxy}ethan-1-ol
1-[2-(1H-imidazol-2-yl)benzoyl]-N-(4-methoxyphenyl)piperidin-3-amine
2-[4-({3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)phenoxy]pyrimidine
1-[(4-methoxyphenyl)methyl]-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
3-(2-{4-[hydroxy(pyridin-2-yl)methyl]piperidin-1-yl}-2-oxoethyl)-1-methyl-3-(4-phenylphenyl)pyrrolidine-2,5-dione
N-{2-[4-(1H-imidazol-4-ylmethyl)morpholin-2-yl]ethyl}-2,2,3,3-tetramethylcyclopropane-1-carboxamide
N-{1-[(5-cyclohexylthiophen-2-yl)methyl]piperidin-3-yl}acetamide
[1-(4-aminopyrimidin-2-yl)-3-[(3-chlorophenyl)methyl]piperidin-3-yl]methanol
methyl 4-[(7-fluoro-3-methyl-1-benzofuran-2-yl)formamido]butanoate
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-methyl-6-{2-[(2-phenylquinazolin-4-yl)amino]ethyl}-3,4-dihydropyrimidin-4-one
1-[(4,5-dimethylfuran-2-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
2-{4-[2-(4-fluorophenyl)-2-hydroxyacetyl]-2-oxopiperazin-1-yl}benzonitrile
3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-[2-(morpholin-4-yl)ethyl]propanamide
3-{3-cyclopentyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-4,5,6,7-tetrahydro-2H-indazole
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-4-methyl-2-oxo-N-(oxolan-2-ylmethyl)pentanamide
methyl({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl})[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
2-[2-(1H-imidazol-4-yl)ethyl]-8-[(5-methylfuran-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-N,N-dimethylpyrimidin-4-amine
2-chloro-N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-5-(trifluoromethyl)benzamide
N,3-diethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-5-hydroxyadamantane-1-carboxamide
N-(2-methylbutyl)-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
2-{4-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]phenoxy}ethan-1-ol
3-(3-methoxyquinoxalin-2-yl)-1-(thiomorpholin-4-yl)propan-1-one
1-{1-ethyl-5-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-4-phenylpiperazine
methyl 2-({4-[1-(3-fluorobenzoyl)piperidin-3-yl]-5-(4-fluorophenyl)pyrimidin-2-yl}sulfanyl)acetate
3,6-dimethyl-N-[1-(thiophen-2-yl)propyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
[(3R,4R)-1-[(2,3-dimethyl-1H-indol-7-yl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-{7-[(4-acetylpiperazin-1-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(2H-1,3-benzodioxol-5-yl)ethan-1-one
4-(1H-imidazol-1-yl)-N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)benzamide
3-[(3R,4S)-1-(1H-indol-5-ylmethyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
5-[2-(ethanesulfinyl)ethyl]-1-(2-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazole
3-[2-(dimethylamino)ethyl]-5-(2-phenylethyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
N-[2-(dimethylamino)-1-phenylethyl]-5-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
7-(1H-1,3-benzodiazol-2-ylmethyl)-N-cyclopropyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N,2-dimethyl-3-{[5-(phenoxymethyl)-1H-pyrazol-3-yl]formamido}propanamide
4-(2,3-dihydro-1H-isoindole-2-carbonyl)-7-methoxy-2-(1H-pyrazol-4-yl)quinoline
2-(2,4-dimethoxyphenyl)-N-ethyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
1-(5-chloropyridin-2-yl)-4-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperazine
3-({1-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]pyrrolidin-3-yl}methyl)benzamide
N-[2-(3-fluorophenyl)ethyl]-1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-1H-1,3-benzodiazole-7-carboxamide
4-methyl-1-({4-[2-(4-methylpiperidin-1-yl)-2-oxoethoxy]phenyl}methyl)piperidine-4-carbonitrile
5,6-dimethyl-3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2-dihydropyridin-2-one