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2-(2,4-dichlorophenoxy)-1-(3-propoxypiperidin-1-yl)ethan-1-one
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
(1R,5R)-6-[2-(benzyloxy)ethyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-{[({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}-5-methoxyphenol
3-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-5-cyclopropyl-1,2-oxazole
N-methyl-1-(2-phenylethyl)-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]piperidin-3-amine
6-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-N,N-dimethylpyridine-3-carboxamide
4-benzyl-1-cyclobutanecarbonyl-3-ethyl-1,4-diazepan-5-one
N-(2-{imidazo[1,2-a]pyrimidin-2-yl}ethyl)-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide
2-(3-methyl-1,2-oxazol-5-yl)-1-(6-methyl-2-phenyl-1,2-diazinan-1-yl)ethan-1-one
2-[2-(1-{2-[(cyclopropylmethyl)sulfanyl]acetyl}piperidin-4-yl)-1H-imidazol-1-yl]acetamide
6-(2,5-dihydro-1H-pyrrol-1-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
(1S,5R)-6-[(2-fluoro-5-methoxyphenyl)methyl]-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(4-fluorophenyl)methyl]-N-[1-(pyridin-2-yl)propan-2-yl]-1H-1,2,3-triazole-4-carboxamide
(1S,5R)-3-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
methyl 1-(benzyloxy)-8-[(6-methyl-4-oxo-4H-chromen-3-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
(3R,4R)-1-[2-(4-fluorophenoxy)ethyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
2-(5-{1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]pyrrolidin-2-yl}-1,2,4-oxadiazol-3-yl)pyridine
3-{2-[1-(2-methoxyphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyridine
2-[1-(3-methoxypropyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)acetamide
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(1-methylpiperidin-4-yl)acetamide
(2R,6R)-10-methoxy-4-[(2-methyl-1,3-thiazol-4-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
{3-[(2,4-difluorophenyl)methyl]-1-[3-(morpholin-4-yl)benzoyl]piperidin-3-yl}methanol
(4-{[3-(2-aminoethyl)phenyl]methyl}-1,4-oxazepan-6-yl)methanol
8-[(2E)-but-2-en-1-yl]-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)methyl]benzonitrile
N-benzyl-7-acetamido-N-(2-hydroxyethyl)-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
(1S,6R)-N-[(3-methoxyphenyl)methyl]-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
N-[4-({ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]carbamoyl}methyl)phenyl]butanamide
ethyl 4-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}piperidine-1-carboxylate
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-[(2-methyl-1,3-oxazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
6-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-propylpyrimidin-4-amine
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-3-(2-methoxyphenyl)propan-1-one
N-ethyl-N-methyl-6-[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})amino]pyridine-3-carboxamide
methyl 7-oxo-3-(2-phenoxyacetyl)-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(2S,3R)-2-amino-1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-hydroxybutan-1-one
N-methyl-N-(oxan-2-ylmethyl)-1,8-naphthyridine-2-carboxamide
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-2-(2,5-dioxo-1-propylimidazolidin-4-yl)acetamide
1-{4-[2-methyl-4-(4-methylphenyl)piperazin-1-yl]-4-oxobutyl}pyrrolidin-2-one
[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl){[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
N-[(2-chlorophenyl)methyl]-3-[1-(2,3-dimethoxybenzoyl)piperidin-3-yl]propanamide
(3S)-1-{2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carbonyl}pyrrolidin-3-ol
2-{1-[(2-fluorophenyl)methyl]-4-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-{3-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-oxopropyl}acetamide
2-({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)-2-methylpropan-1-ol
4-[2-(4-fluoro-2-methylphenyl)acetyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
3-(cyclopropylmethyl)-5-(oxolan-3-yl)-1-[4-(trifluoromethoxy)phenyl]-1H-1,2,4-triazole
2-{[4-(4-methylphenyl)-5-(piperidin-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
1-{3-[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-oxopropyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one