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3-(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)-1-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}urea
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-(pentan-3-yl)piperazin-2-yl}ethan-1-ol
2-methyl-3-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,8-naphthyridine
2,5-dimethyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}pyrimidin-4-amine
(2R,6R)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
5-{1-[(2Z)-2-fluoro-3-phenylprop-2-enoyl]piperidin-4-yl}-5-[(4-fluorophenyl)methyl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
N-(furan-2-ylmethyl)-3-(1-phenylethyl)-N-(prop-2-yn-1-yl)-1,2-oxazole-5-carboxamide
2-(5-acetylthiophen-3-yl)-1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]ethan-1-one
1-[(4-ethylphenyl)methyl]-4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]piperidine
3-[(3,5-dimethylphenyl)methyl]-9-methoxy-7-oxo-N-[3-(1H-pyrazol-1-yl)propyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-amino-6-cyclopropyl-4-[2-(2-hydroxyethoxy)phenyl]pyridine-3-carbonitrile
4,6-dimethyl-3-[4-(pyridin-4-yloxy)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-(propan-2-yl)-4-[3-(pyridin-2-yl)propanoyl]-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
1-(2-{[(4-chlorophenyl)methyl]amino}ethyl)-N-(3-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide
2-methoxy-1-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
8-[4,5-dimethyl-2-(1H-pyrrol-1-yl)thiophene-3-carbonyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
{3-[2-(1-phenyl-1H-pyrazol-5-yl)-1H-imidazol-1-yl]phenyl}methanol
7-(cyclohexylmethyl)-2-(thiophene-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(3S,4S)-1-[(2-chloro-4,5-dimethoxyphenyl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
1-[(4-fluorophenyl)methyl]-N-methyl-N-{[4-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
(3S,4R)-4-phenyl-1-(2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}acetyl)pyrrolidine-3-carboxylic acid
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(5-hydroxypyrazine-2-carbonyl)piperazin-2-one
2-{5-[(E)-2-(4-fluorophenyl)ethenyl]-4-phenyl-1H-imidazol-1-yl}-1-(pyridin-3-yl)ethan-1-ol
1-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-4-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-1,2,3-triazole
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-[(4-fluorophenyl)methyl]propanamide
6-methoxy-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-[1-(2,6-difluorobenzoyl)piperidin-3-yl]-2-methyl-5-(3-methylphenyl)pyrimidine
{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}(pyridin-3-ylmethyl)amine
2,6-dimethyl-N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}quinoline-4-carboxamide
1-(2-methoxyphenyl)-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
N-[2-(4-{[(2,2-diethylcyclopropyl)formamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]pyridine-3-carboxamide
(1R,5R)-6-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
6-{[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(3-chlorophenyl)-4-[4-(propan-2-yloxy)benzoyl]piperazin-2-one
N-(furan-2-ylmethyl)-3-{[3-(2-hydroxyethoxy)phenyl]methyl}-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N5-cyclooctyl-4-oxo-N3,N3-bis(prop-2-en-1-yl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
ethyl 4-[(2S,4S)-4-[4-(methoxycarbonyl)-1H-1,2,3-triazol-1-yl]-2-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-1-yl]piperidine-1-carboxylate
7-amino-4-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
1-{5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-3-ol
1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-2-[1-(propan-2-yl)piperidin-4-yl]ethan-1-one
1-[(2,3-difluorophenyl)methyl]-4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
(4aR,7aS)-1-(2-methoxyethyl)-4-(2,2,3,3-tetramethylcyclopropanecarbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1R,7S)-3-[(3-methoxyphenyl)methyl]-6-(morpholine-4-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
2-{4-[2-hydroxy-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]morpholin-3-yl}-1-(pyrrolidin-1-yl)ethan-1-one
3-(4-chlorobenzoyl)-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidine
1-{3-[3-(3-hydroxypropyl)-4H-1,2,4-triazol-4-yl]phenyl}ethan-1-one
methyl (2S)-1-[3-(2,5-difluorobenzoyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl]pyrrolidine-2-carboxylate
3-(but-2-yn-1-yl)-5-(2-phenylethyl)-5-[1-(3-phenylpropyl)piperidin-4-yl]imidazolidine-2,4-dione
N-methyl-N-{2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}-4-(trifluoromethyl)benzene-1-sulfonamide
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(2-phenylethyl)acetamide