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ethyl 3-[(4-fluorophenyl)methyl]-1-[3-(4-fluorophenyl)propanoyl]piperidine-3-carboxylate
2-[4-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
3-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-1-(2,4,6-trimethylpyridin-3-yl)urea
3-{1-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)propanamide
methyl (2R)-2-{[(2S,4S)-4-cyclohexaneamido-1-methylpyrrolidin-2-yl]formamido}propanoate
2-{[(5-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}ethan-1-ol
4-(hydroxymethyl)-1-[(6-methylquinolin-5-yl)methyl]azepan-4-ol
N-cyclopropyl-2-(2-hydroxyphenyl)-N-[(2-methoxyphenyl)methyl]acetamide
1-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(furan-2-yl)ethane-1,2-dione
N-[(2-chlorophenyl)methyl]-3-(1-phenylethyl)-1,2-oxazole-5-carboxamide
N-[2-(4-chlorophenyl)ethyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-N-(1-methanesulfonylpiperidin-4-yl)propanamide
6-fluoro-4-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazine-1-carbonyl}-1,2,3,4-tetrahydroquinolin-2-one
N-(2,2-dimethyloxan-4-yl)-1-[1,3-dioxo-2-(quinolin-3-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carboxamide
3-{1-[3-(3-fluorophenyl)propanoyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
1-(4-{[(2,1,3-benzoxadiazol-5-ylmethyl)amino]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
(1R,3S,5S)-8-[6-methyl-2-(morpholin-4-yl)pyrimidin-4-yl]-8-azabicyclo[3.2.1]octan-3-ol
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
2-fluoro-4-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenol
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(propan-2-yl)-1-{[4-(propan-2-yl)phenyl]methyl}pyrrolidine-2-carboxamide
1-(2-methoxyacetyl)-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-2-fluoro-5-sulfamoylbenzamide
N-[2-(azepan-1-yl)-2-phenylethyl]-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
2-(4-fluorophenyl)-N-[2-(7-{[2-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]acetamide
6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-1,4-diazepan-2-one
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-6-(methoxymethyl)pyrimidin-4-amine
2,6-dimethyl-N-[1-(pyrrolidin-1-ylmethyl)cyclohexyl]pyridine-4-carboxamide
N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)cyclohex-3-ene-1-carboxamide
1-cyclohexyl-N-cyclopropyl-5-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
1-methyl-4-[(2S,4R)-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidine-2-carbonyl]-1,4-diazepane
N-[2-(azepan-1-yl)ethyl]-3-(4-hydroxyphenyl)-N-methylbenzamide
(1R,4S)-1,7,7-trimethyl-3-oxo-N-(4H-1,2,4-triazol-4-yl)-2-oxabicyclo[2.2.1]heptane-4-carboxamide
5-benzamido-1-cyclopentyl-N-[2-(1H-pyrazol-4-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
1-[6-methyl-3-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)quinolin-2-yl]piperidin-3-ol
(3aS,7aR)-5-methyl-2-{2-[3-(trifluoromethyl)phenyl]acetyl}-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
N-cyclopropyl-2-[(2,3-dimethoxyphenyl)methyl]benzamide
2-({[(1R,3R)-3-aminocyclopentyl]amino}methyl)-8-fluoroquinolin-4-ol
N-methyl-N-[2-(morpholin-4-yl)propyl]-2-(4-propanoylphenoxy)acetamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopropyl-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2-(2-{[1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)-6-methyl-3,4-dihydropyrimidin-4-one
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(methylsulfanyl)benzamide
2-cyclopentyl-N-methyl-N-{2-[4-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenoxy]ethyl}acetamide
1-{4-[(4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)methyl]thiophen-2-yl}ethan-1-one
7-fluoro-3-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-1-(oxolan-2-ylmethyl)-1,2-dihydroquinolin-2-one
3-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(cyclohex-1-en-1-ylmethyl)-3-(8-fluoro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea
3-(2-fluorophenoxy)-1-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}azetidine
(2,1,3-benzoxadiazol-5-ylmethyl)[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl]methylamine
methyl 3-{[3-(3,4-dimethoxyphenyl)propanamido]methyl}-5-[2-(thiophen-3-yl)acetamido]benzoate