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1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
(3S,4R)-1-(isoquinoline-5-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
ethyl 2-(4-{[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}morpholin-3-yl)acetate
N-(2,1,3-benzoxadiazol-5-ylmethyl)-6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-oxo-1-(2-phenylethyl)piperidine-3-carboxamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-(1-phenylethyl)benzamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-ol
4-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-methoxypyridine-3-carbonitrile
5-cyclopropyl-N-[2-(diethylamino)ethyl]-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-N-methyl-1H-pyrazole-4-carboxamide
1-{4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}-4-(2-methylphenyl)piperazine
1-[6-(2,6-dimethoxypyridin-3-yl)pyridin-2-yl]ethan-1-ol
2-amino-6-[1-(3-chlorophenyl)-1H-pyrazol-4-yl]-4-(pyridin-3-yl)pyridine-3-carbonitrile
N-ethyl-2-methyl-N-[3-(morpholin-4-yl)propyl]-2-(thiophen-2-ylformamido)propanamide
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-(1-phenylcyclopropyl)acetamide
2-(4-methylpyrimidin-2-yl)-9-oxa-2-azaspiro[5.5]undecane
8-[(1-ethyl-1H-pyrazol-3-yl)methyl]-8-azaspiro[4.5]decane-7,9-dione
2-[(4-chlorophenyl)methyl]-8-(5-ethyl-1,2,4-oxadiazol-3-yl)-2,8-diazaspiro[4.5]decan-3-one
4-{2-[3-(2-methoxybenzoyl)piperidin-1-yl]-2-oxoethyl}-7-methyl-2H-chromen-2-one
4-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-1-(3-methoxyphenyl)piperazin-2-one
3-chloro-4-({1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
3-{5-[({[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}amino)methyl]thiophen-3-yl}prop-2-yn-1-ol
N-(1,4-dioxan-2-ylmethyl)-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
1-(2-methoxyethyl)-1-(1-methylpiperidin-4-yl)-3-[2-(pyridin-3-yloxy)phenyl]urea
2-{4-[(dimethylamino)methyl]-4-hydroxyazepane-1-carbonyl}-5-methoxy-4H-pyran-4-one
1-[1'-(2,3-dihydro-1-benzofuran-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
6-(cyclopropylmethoxy)-4-(2,3-difluorobenzoyl)-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3,4,5-trimethoxyphenyl)acetamide
2-acetamido-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]acetamide
6-methyl-2-[1-(morpholine-4-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
2,4-difluoro-3-methoxy-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methylbenzamide
(4aR,8aS)-1-(3-ethoxypropyl)-6-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-decahydro-1,6-naphthyridin-2-one
1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-[methyl(phenyl)amino]ethan-1-one
5-({3-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)isoquinoline
1-benzyl-8-(3-phenylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(oxolan-3-ylmethyl)-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine
3-({[1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-4-yl]oxy}methyl)pyridine
1-methyl-2-oxo-N-[3-(propan-2-yloxy)propyl]-1,2-dihydropyridine-4-carboxamide
2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}-N-[(1r,4r)-4-hydroxycyclohexyl]acetamide
methyl 6-(1-methylcyclopropanecarbonyl)-2-[(2-phenylethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-methoxy-1-{1'-[(2-methylphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-2-(pyridin-2-yl)pyrimidine-5-carboxamide
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-3-carboxamide
(3S,4S)-1-(6-methylpyridine-2-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
(2S,4R)-4-amino-1-[(2S)-2-methoxy-2-phenylacetyl]-N-methylpyrrolidine-2-carboxamide
2-{2-cyclopropyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-N,N-dimethylacetamide
8-(furan-3-carbonyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
3-{[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}-3-(4-methylphenyl)propan-1-ol
N-{[3-(cyclopentyloxy)-4-methoxyphenyl]methyl}-4-(4-methylphenyl)-N-(pyridin-4-ylmethyl)benzamide
3-(3-methylthiophene-2-carbonyl)-1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidine
N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-3-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide