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2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[1-(3-methoxyphenyl)ethyl]-N-methylacetamide
2-(oxolan-3-ylmethyl)-1H,2H,3H,4H,5H-pyrido[4,3-b]indole
N-cyclopropyl-2-{9-oxo-8-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-2-yl}acetamide
3-[(benzylamino)methyl]-5-acetamido-N-(4-methoxyphenyl)benzamide
{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}({[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl})amine
2-[4-(cyclohex-3-ene-1-carbonyl)piperazin-1-yl]-1,3-benzothiazole
1-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-3-propylurea
3-[2-oxo-2-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethyl]-1,3-oxazolidin-2-one
5-acetamido-1-(2-methoxyethyl)-N-[2-(4-methylphenyl)ethyl]-2-(pyridin-2-yl)-1H-1,3-benzodiazole-7-carboxamide
3-(1,3-benzothiazol-2-yl)-N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)propanamide
[(3R,4R)-1-(9H-fluorene-9-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]-2,3-dimethylquinoxaline-6-carboxamide
methyl 9-{2-cyano-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-3-azaspiro[5.5]undecane-3-carboxylate
3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-(4-methyl-4-phenylpentan-2-yl)propanamide
4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-6-(piperidin-1-yl)pyrimidine
N-butyl-N-methyl-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
2-butanoyl-7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decan-6-one
2-[1-cyclohexyl-4-(3-phenylpropyl)piperazin-2-yl]ethan-1-ol
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
(2S)-2-amino-1-(4-{[(4-fluorophenyl)methyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)-3-hydroxypropan-1-one
N-(5-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}pyrimidin-2-yl)benzenesulfonamide
2-(dimethylamino)-2-(3-fluorophenyl)-1-{4-[2-(1H-pyrrol-1-yl)ethyl]piperazin-1-yl}ethan-1-one
6-chloro-1-methyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1H-indole-2-carboxamide
2-[(7-chloro-1-methyl-1H-indol-2-yl)formamido]-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetic acid
1-[2-(propan-2-ylsulfanyl)phenyl]-3-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}urea
methyl[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)amine
2-[5-(4-methylbenzoyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline
1-methyl-4-[(3-methyl-1,2-benzoxazol-5-yl)methyl]piperazine-2-carboxylic acid
1-{4-[3-(3-methoxypropyl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
N-[3-(azepan-1-yl)propyl]-3-ethyl-N-methyl-1H-indole-2-carboxamide
3-({6-oxo-1-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}methyl)-2,3-dihydro-1,3-benzoxazol-2-one
1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-4-methylpentane-1,2-dione
methyl 2-(cyclopentylsulfamoyl)-6-[(2E)-2-methylbut-2-enoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-ethyl-4-(pyrrolidin-1-ylmethyl)-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]furan-2-carboxamide
ethyl 4-[2-(phenylamino)pyrimidine-5-amido]piperidine-1-carboxylate
5-methyl-N-({1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperidin-3-yl}methyl)-1,2-oxazole-3-carboxamide
7-chloro-2-{[4-(4-methylphenyl)piperazin-1-yl]methyl}-4-(morpholin-4-yl)quinazoline
2-{2-[(4,4,4-trifluorobutan-2-yl)amino]ethyl}-1,2,3,4-tetrahydrophthalazine-1,4-dione
1-ethyl-N-[(5-methylpyrazin-2-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-1-[2-(trifluoromethyl)phenyl]urea
2-(2-methyl-1,3-thiazol-4-yl)-1-[3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethan-1-one
N-[3-(3-chlorophenyl)phenyl]-1-(furan-3-carbonyl)piperidine-4-carboxamide
2-[4-(3-methoxybenzoyl)piperazine-1-carbonyl]pyrrolidine-1-carboxamide
{[2-(azocan-1-yl)pyridin-3-yl]methyl}({[5-(methoxymethyl)furan-2-yl]methyl})amine
11-{[(3,5-difluorophenyl)methyl]amino}-4-[2-(morpholin-4-yl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
methyl 4-{[1-benzyl-3-(3-oxopiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}benzoate
1-[2-(3-fluorophenyl)ethyl]-6-oxo-N-(propan-2-yl)piperidine-3-carboxamide
(3S,4R)-1-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
3-{2-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-2-oxoethyl}-4-(2-phenylethyl)piperazin-2-one
N-[(4-cyanophenyl)methyl]-1-(oxan-4-yl)piperidine-4-carboxamide