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3-[2-(4-methoxyphenyl)ethyl]-1-(propane-1-sulfonyl)piperidine
3-{1-[(9-ethyl-9H-carbazol-3-yl)methyl]piperidin-3-yl}-1-(morpholin-4-yl)propan-1-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(1-benzylpiperidin-3-yl)methyl]acetamide
methyl 2-{[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl](methyl)amino}acetate
(3S,9aR)-3-(1H-imidazol-4-ylmethyl)-8-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(2S)-2-(methoxymethyl)-N-(quinolin-3-yl)pyrrolidine-1-carboxamide
2-benzyl-8-(pyrazin-2-yl)-2,8-diazaspiro[5.5]undecane
2-{[(1R,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}quinolin-4-ol
N-(4-{[1-(2-methoxyethyl)-2,4-dioxo-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decan-8-yl]methyl}phenyl)acetamide
methyl 3-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-7-oxo-9-[2-(piperidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(5S)-5-({[(1-phenyl-1H-pyrazol-4-yl)methyl](pyridin-3-ylmethyl)amino}methyl)pyrrolidin-2-one
N-[(2R,3R)-1'-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxyacetamide
N-(3-fluorophenyl)-6-[(4-methoxy-3-methylphenyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}(1,4-dioxan-2-ylmethyl)amine
N-[(3R,4S)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-propylpyrrolidin-3-yl]-2-methoxyacetamide
4-[(3-fluorophenyl)methyl]-1-[2-(thiophen-3-yl)acetyl]-1,4-diazepan-5-one
N-(3-hydroxypropyl)-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
N-(1-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N-ethyloxane-4-carboxamide
3-({2-ethyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}methyl)benzonitrile
3-{3-[({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}amino)methyl]-1H-indol-1-yl}propanamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]acetamide
5-fluoro-2-(1-{1-[4-(morpholine-4-carbonyl)phenyl]piperidin-4-yl}piperidin-4-yl)-1H-1,3-benzodiazole
2-methoxy-1-(4-{[4-(pyridin-2-yl)phenyl]methyl}-1,4-diazepan-1-yl)ethan-1-one
2-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-6-methylpyridine-3-carbonitrile
3-[3-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]benzonitrile
methyl (2S)-2-{[1-(7-methoxy-4-methylquinazolin-2-yl)piperidin-4-yl]formamido}-3-methylbutanoate
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}(pyridin-3-ylmethyl)amine
(4aS,8aS)-2-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-decahydroisoquinolin-4a-ol
1-[2-(4-methoxyphenyl)ethyl]-3-(2-methylpropyl)-8-(1,2,3,4-tetrahydronaphthalen-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N,N-diethyl-3-(1-methyl-1H-indazol-5-yl)benzamide
methyl (2S,4S,5R)-5-(2-chlorophenyl)-1,2-dimethyl-4-{[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]carbamoyl}pyrrolidine-2-carboxylate
ethyl 1-(2-methylphenyl)-5-[(4-methylpiperazin-1-yl)methyl]-1H-pyrazole-4-carboxylate
1-ethyl-6-methyl-3-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
(5S,9aS,9bS)-2-cyclopentyl-5-[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-methyl-8-[(2-methylphenyl)methyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
7-{2-[2-(trifluoromethyl)phenyl]acetyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)cyclopentanecarboxamide
6-[(3-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-[3-(2-oxoimidazolidin-1-yl)benzoyl]-1,4-diazepan-2-one
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
2-(2,6-dimethoxyphenyl)pyridine-3-carbonitrile
8-fluoro-N-[1-(phenylcarbamoyl)piperidin-4-yl]quinoline-2-carboxamide
3-[4-(3-methylphenyl)piperazin-1-yl]-N-(pyridin-3-ylmethyl)propanamide
2-[(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidin-4-yl)oxy]pyrimidine
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl][2-(pyridin-3-yloxy)propyl]amine
1-cyclopropyl-N-methyl-5-oxo-N-(quinoxalin-2-ylmethyl)pyrrolidine-3-carboxamide
N-methyl-1-(piperidin-3-ylmethyl)-N-(1,3-thiazol-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
({3-[(1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-4-yl)oxy]phenyl}methyl)(furan-3-ylmethyl)methylamine
N'-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-N-(propan-2-yl)ethanediamide
N-(1-cyclohexyl-1H-pyrazol-5-yl)-2-(4,5-dichloro-1H-imidazol-1-yl)acetamide