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1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
5-(4-methoxyphenyl)-N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}furan-2-carboxamide
2-(dimethylamino)-2-(4-fluorophenyl)-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}acetamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-5-cyclopropyl-1,3,4-oxadiazol-2-amine
7-[(2-fluorophenyl)methyl]-2-[(1-methyl-1H-imidazol-2-yl)methyl]-2,7-diazaspiro[4.5]decane
3-(dimethylamino)-N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)benzamide
2-(3-{[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)quinoxaline
methyl 5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxylate
(2S,4S)-4-[(cyclohexylmethyl)amino]-1-{[4-(diethylamino)phenyl]methyl}-N-methylpyrrolidine-2-carboxamide
N-methyl-N-(1,2-oxazol-5-ylmethyl)-3-(1H-pyrazol-1-yl)benzamide
N3-[2-(3-methoxyphenoxy)ethyl]-N1,N1,N3-trimethylpiperidine-1,3-dicarboxamide
N-(2-hydroxyethyl)-5-{[(4-methylphenyl)carbamoyl]carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
8-[(4-carbamoylphenyl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-phenyl-N-{2-[3-(thiomorpholin-4-ylmethyl)phenoxy]propyl}benzamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)acetamide
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]propanamide
5-{[3-(2-ethoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-2-(furan-2-yl)pyrimidine
1-{6-azabicyclo[3.2.1]octan-6-yl}-2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
N,N-dimethyl-4-{3-[methyl(2-phenylethyl)amino]piperidine-1-carbonyl}piperidine-1-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)-1,4-diazepane
4-(2,6-dimethylpyridin-3-yl)-N-[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]pyrimidin-2-amine
(3S,9aR)-3-ethyl-8-(thiophen-2-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}ethan-1-one
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]pyrrolidin-3-yl]methanol
(3S,4S)-1-[2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetyl]-4-propylpyrrolidine-3-carboxylic acid
5-cyclopropanecarbonyl-1'-(1-ethyl-1H-pyrazole-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N,N-diethyl-1-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperidine-3-carboxamide
2,3-dimethoxy-N-{[1-(thian-4-yl)piperidin-3-yl]methyl}benzamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(5-methyl-1,3-oxazole-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
3-(1H-imidazol-1-ylmethyl)-1-[5-(3-methoxyphenyl)furan-2-carbonyl]piperidine
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
3-ethyl-8-{[4-(2-hydroxyethoxy)phenyl]methyl}-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(methylsulfanyl)acetamide
5-({[2-(4-chlorophenyl)ethyl]carbamoyl}methyl)-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-ethyl-N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
4-(1H-1,3-benzodiazol-1-yl)-1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxylic acid
5-methyl-5-{1-[1-methyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carbonyl]piperidin-4-yl}imidazolidine-2,4-dione
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-(6-methylpyridine-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
5-(1-ethyl-1H-imidazol-2-yl)-1-[(2-methoxyphenyl)methyl]-4-phenyl-1H-imidazole
1-methyl-3-(propan-2-yl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[(3S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-1-(morpholin-4-yl)propan-1-one
1'-(5-acetyl-2,4-dimethyl-1H-pyrrole-3-carbonyl)-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-[(4-methyl-1,4-diazepan-1-yl)sulfonyl]-N-(1,2-oxazol-3-ylmethyl)benzamide
N-(2-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}-1,2,3,4-tetrahydroisoquinolin-7-yl)oxolane-2-carboxamide
{5-[(3-chloropyridin-4-yl)methyl]-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
3-[1-(1-cyclobutanecarbonylpiperidine-4-carbonyl)azetidin-3-yl]pyridine
1-[1-(cyclopropylmethyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-4-carboxamide
1-(furan-2-yl)-2-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]ethane-1,2-dione
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-methyl-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}urea
1-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-3-methylpentan-1-one