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2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]-1-(3-methylpiperidin-1-yl)ethan-1-one
2-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}-4-phenyl-1,3-thiazole
2-{[5-(5-ethylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-5-methyl-1,3,4-oxadiazole
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}propanamide
(4aS,7aR)-4-[(4-chlorophenyl)methyl]-N-ethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-(3-phenylpropyl)piperidin-4-ol
2-{1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-1,2,3,4-tetrahydroisoquinoline
(5-{[1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
2-[4-(1,4-dithiepan-6-yl)-1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-({5-[(cyclohexylmethyl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}methyl)-3-(3,5-dimethyl-1H-pyrazol-1-yl)propanamide
2-(2-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-4-(morpholin-4-yl)pyrimidin-5-yl)-2-methylpropanoic acid
4-methyl-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}pyrimidin-2-amine
1-[1-(2-methoxypyridine-4-carbonyl)piperidin-4-yl]piperidin-3-ol
2-{[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
8-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
4-[(1R,9aR)-octahydro-1H-quinolizine-1-carbonyl]-1-(2-methoxyphenyl)piperazin-2-one
2-[5-(2-benzyl-1,3-thiazole-4-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
1-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinolin-8-yl)-3-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}urea
4-benzyl-4-(hydroxymethyl)-N-[3-(trifluoromethyl)phenyl]piperidine-1-carboxamide
2-ethyl-1-[(4-methoxyphenyl)methyl]-6-methyl-4-oxo-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}-1,4-dihydropyridine-3-carboxamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1-(propan-2-yl)piperidine
1-[(2-phenyl-1H-imidazol-4-yl)methyl]-4-propylpiperazine
5-[2-(methylsulfanyl)propyl]-4-phenyl-1-[(1-propyl-1H-imidazol-2-yl)methyl]-1H-imidazole
2-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]thiophen-3-amine
2-{[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]amino}pyridine-3-carbonitrile
7-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[2-(propan-2-yloxy)ethyl]benzamide
1-({1-[6-(dimethylcarbamoyl)pyrazin-2-yl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxylic acid
2-(4-aminopyrimidin-2-yl)-7-cyclopentyl-2,7-diazaspiro[4.5]decan-6-one
1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
2-methoxy-1-{3-[4-(4-methylphenyl)piperazine-1-carbonyl]piperidin-1-yl}ethan-1-one
(4aR,8aS)-6-(2-fluorobenzoyl)-1-(1-methyl-1H-pyrazole-5-carbonyl)-decahydro-1,6-naphthyridine
3-(4-methyl-1,3-thiazol-5-yl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]propanamide
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(furan-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)acetamide
2-{[3-(2-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-methyl-1H-1,3-benzodiazole
3-(4-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)-2,5-dimethylpyrazine
1-(2-amino-6-methylpyrimidin-4-yl)-4-(1H-pyrrole-2-carbonyl)-1,4-diazepane-6-carboxylic acid
N-[(3-methoxyphenyl)methyl]-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
5-cyclopentanecarbonyl-3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
7-acetamido-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
1-(3-fluoropyridin-2-yl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
3-(5-{5-[(methylsulfanyl)methyl]furan-2-yl}-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl)pyridine
3-methyl-8-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
4-[2-(3-methoxyphenyl)phenyl]-4H-1,2,4-triazole
N,3,6,7-tetramethyl-N-[1-(pyridin-2-yl)propyl]-1-benzofuran-2-carboxamide
[4-({4-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-1H-1,2,3-triazol-1-yl}methyl)oxan-4-yl]methanol
4-(3-fluorophenoxy)-1-(4-methoxypyrimidin-2-yl)piperidine-4-carboxylic acid
2-chloro-4-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)phenol
2-(4-chlorophenyl)-4-[5-(propan-2-yl)pyrimidin-4-yl]morpholine