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N-[3-(1H-indol-2-yl)phenyl]-1-(oxolan-3-ylmethyl)piperidine-4-carboxamide
N-{1-[1-(quinolin-8-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
N-[2-(diethylamino)ethyl]-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carboxamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-[2-(2-methoxyphenyl)ethyl]benzamide
1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-1,4-diazepane-6-carboxylic acid
1-(2-chloroprop-2-en-1-yl)-3-[(cyclopropylamino)methyl]-6,7-dimethoxy-1,2-dihydroquinolin-2-one
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
6-chloro-N,N-dimethyl-2-(1-propyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
2,6,8-trimethyl-4-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]quinoline
8-[(5-chloro-2-hydroxyphenyl)methyl]-1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-(1-ethylpiperidin-4-yl)acetamide
methyl 4-(5-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
1-cycloheptyl-N-methyl-N-(oxan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-(1H-indol-3-yl)-N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]acetamide
N-methyl-2-(methylsulfanyl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
5-[1-(3-cyclohexylpropanoyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
(2S)-N-(3-chloro-2-fluorophenyl)-2-(methoxymethyl)pyrrolidine-1-carboxamide
4-{4-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]-2-oxopiperazin-1-yl}benzonitrile
4-[5-(2,3-dichlorophenyl)furan-2-yl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-{1'-[(2S)-1-acetylpyrrolidine-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
2-methyl-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}imidazo[1,2-a]pyrimidine-3-carboxamide
(2R)-2-amino-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-2-phenylacetamide
2-methoxy-N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-phenylacetamide
6-(benzyloxy)-4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
ethyl 1-[5-(methoxymethyl)furan-2-carbonyl]-4-(3-phenylpropyl)piperidine-4-carboxylate
(1S,5R)-6-(cyclopropylmethyl)-3-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N,N-diethyl-2-({4-[1-(2-methoxyethyl)-5-oxopyrrolidine-3-carbonyl]-2-oxo-1-(2-phenylethyl)-1,4-diazepan-6-yl}oxy)acetamide
2-[(1-acetylpiperidin-4-yl)oxy]-N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-5-methoxybenzamide
7-(5-propyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-6-methylphenol
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-[4-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide
({5-[1-(2,3-dihydro-1-benzofuran-5-carbonyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
methyl (2S,4R)-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamido]-1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]pyrrolidine-2-carboxylate
N4-[3-(2-amino-1,3-thiazol-4-yl)propyl]-5-ethylpyrimidine-2,4-diamine
(3S,4S)-4-cyclopropyl-1-[(5-ethylfuran-2-yl)methyl]pyrrolidine-3-carboxylic acid
2-{[2-(2,3-difluoro-6-methoxyphenyl)-1H-imidazol-1-yl]methyl}-5-ethylpyridine
3-(benzyloxy)-1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
4-[2-(3,5-dimethoxyphenyl)acetyl]-1-ethyl-3-methylpiperazin-2-one
N-methyl-N-[(3-methylthiophen-2-yl)methyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[1-(2-hydroxyethyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
{4-benzyl-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}methanol
1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(3-methylphenoxy)piperidine
ethyl 4-(2-phenoxyethyl)-1-[3-(1H-1,2,4-triazol-1-yl)propanoyl]piperidine-4-carboxylate
1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-4-[(4-methylphenyl)methyl]-1,4-diazepan-5-one
2-[(5-methyl-1-propyl-1H-pyrazol-4-yl)formamido]-N-(1,3-thiazol-2-yl)acetamide
N-(1H-imidazol-2-ylmethyl)-1-[(2-methoxyphenyl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[3-(2-oxo-2-{4-[2-(pyridin-4-yl)ethyl]piperazin-1-yl}ethoxy)phenyl]propanamide
2-methoxy-N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]acetamide
2-{benzyl[(1,4-dimethyl-1H-pyrazol-5-yl)methyl]amino}ethan-1-ol