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[3-(2-phenylethyl)-1-(thiophene-2-carbonyl)piperidin-3-yl]methanol
4-{5-[1-(furan-2-ylmethyl)piperidin-4-yl]-1,2,4-oxadiazol-3-yl}pyridine
(1S,5R)-3-benzyl-6-[2-methyl-2-(morpholin-4-yl)propyl]-3,6-diazabicyclo[3.2.2]nonane
(3S,4S)-1-[3-(1H-pyrazol-1-yl)propyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
1-(diethylamino)-3-{2-methoxy-5-[(4-methylpiperazin-1-yl)methyl]phenoxy}propan-2-ol
5-benzyl-1-(4-methylphenyl)-4-(1H-pyrrole-2-carbonyl)piperazin-2-one
5-acetyl-6-methyl-3-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2-{[(2R,3S,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}-3,5-dimethyl-1,4-dihydropyridin-4-one
1-{2-[(3,4-dimethoxyphenyl)formamido]ethyl}-N-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
methyl 1-[1-(4-methylquinazolin-2-yl)piperidine-4-carbonyl]piperidine-4-carboxylate
3-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-4-yl}-1-(4-phenylpiperazin-1-yl)propan-1-one
6-[(3-methoxyphenyl)methoxy]-1-(pyridin-2-ylmethyl)-4-[2-(thiophen-2-yl)acetyl]-1,4-diazepan-2-one
N-[2-(cyclohexylsulfanyl)ethyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
4-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}acetamide
2-(3-{[3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]methyl}phenyl)-6-propyl-3,4-dihydropyrimidin-4-one
2-methoxy-1-{1'-[2-(pyridin-4-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
methyl (2S,4S)-4-cyclohexaneamido-1-[(3-fluorophenyl)methyl]pyrrolidine-2-carboxylate
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]({[2-(4-fluorophenyl)-6-methylquinolin-3-yl]methyl})amine
2-[(3-chloro-4,5-dimethoxyphenyl)methyl]-octahydro-1H-pyrido[1,2-a]piperazine
1-[(4-methoxyphenyl)methyl]-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
2-(1,4-dimethylpiperazin-2-yl)-1-{4-[(3-hydroxyphenyl)methyl]piperazin-1-yl}ethan-1-one
1-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}cyclopropan-1-amine
1-[2-(4-chlorophenyl)ethyl]-N-(1H-indol-2-ylmethyl)-6-oxopiperidine-3-carboxamide
3-[3-cyclopropyl-1-(3-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl]-4-methoxybenzene-1-sulfonamide
(3E)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)hex-3-enamide
2-(4-fluorophenyl)-N-(2-{7-[(4-hydroxy-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
N-[2-(4-chlorobenzenesulfonamido)ethyl]-2-(1H-1,2,4-triazol-5-yl)benzamide
N-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-methylpropanamide
1-{1,5-bis[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
N-cyclopropyl-3-{1-[2-(2,6-difluorophenyl)acetyl]piperidin-4-yl}propanamide
2,3-dimethyl-7-[2-(1H-pyrazol-1-yl)propanoyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-{3-[(3S,4S)-3-hydroxy-4-(4-methanesulfonylpiperazin-1-yl)pyrrolidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
2-amino-1-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethan-1-one
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-1-[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]ethan-1-one
[(1-cyclohexylpiperidin-3-yl)methyl][(2-fluoro-4-methoxyphenyl)methyl](pyridin-3-ylmethyl)amine
1,5,6-trimethyl-3-{4-[2-(morpholin-4-yl)ethyl]piperazine-1-carbonyl}-1,2-dihydropyridin-2-one
5-(2,6-difluorophenoxymethyl)-N-(2,3-dihydro-1H-inden-1-yl)-1,2-oxazole-3-carboxamide
1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-3-(trimethyl-1H-pyrazol-1-yl)propan-1-one
8-[(2S)-2,3-dihydroxypropyl]-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
3-{6-[(2-hydroxyethyl)(methyl)amino]pyridazin-3-yl}-5-[2-(piperidin-2-yl)ethyl]phenol
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-methanesulfonyl-2-{[4-methyl-2-(propan-2-yl)-1,3-thiazol-5-yl]formamido}butanoic acid
4-({3-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)piperazin-2-one
N-(1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}pyrrolidin-3-yl)acetamide
methyl 3-(2-chlorobenzoyl)-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-{4-[(4-hydroxyquinolin-2-yl)methyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
5-(2,3-dihydro-1,4-benzodioxin-6-yl)-N,N-dimethylfuran-2-carboxamide
2-[3-(2-chlorophenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]acetamide