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{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
methyl 3-[(3S,4R)-1-(thiophen-2-ylmethyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanoate
N-{[5-(3,6-dimethylpyrazin-2-yl)-7-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-acetamido-3-methylbutanamide
[(5-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
4-{3-[(4,4-dimethylpiperidin-1-yl)methyl]-8-methylimidazo[1,2-a]pyridine-2-carbonyl}morpholine
5-[3-(4-benzylpiperidin-1-yl)-3-oxopropyl]-5-[(2-fluoro-4-methoxyphenyl)methyl]pyrrolidin-2-one
2-(2-methyl-1,3-thiazol-4-yl)-N-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]acetamide
1-(3-methylbutyl)-8-[3-(5-methylfuran-2-yl)butyl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(3-chloro-2-propoxyphenyl)-3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]urea
2-(4-methyl-1,2,5-oxadiazol-3-yl)-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}acetamide
4-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-2-(2-phenylethyl)morpholine
(4S)-4-acetamido-4-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]butanamide
N-cyclopropyl-N-(1-{1-[(2-fluorophenyl)methyl]piperidin-4-yl}-2-phenylethyl)furan-2-carboxamide
N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
2-[1-ethyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
4-({[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]amino}methyl)-N-methylbenzamide
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-(5-methylthiophen-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(4aS,8aR)-1-(2-aminoethyl)-6-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
2-benzyl-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-2-(phenylsulfanyl)ethan-1-one
3-(cyclobutylsulfamoyl)-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]benzamide
3-{1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]piperidin-3-yl}-N-(4-fluoro-2-methylphenyl)propanamide
3-(3-fluorophenyl)-4-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]piperazin-2-one
3-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]-1-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]urea
5-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-4-methyl-2-(pyridin-3-yl)pyrimidine
2-amino-6-(furan-2-yl)-4-[1-(pyridin-2-yl)-1H-pyrrol-2-yl]pyridine-3-carbonitrile
2-[({1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}oxy)methyl]pyridine
(4aS,7aR)-1-(2,2-diphenylacetyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[5-(pyrimidin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1-(pyrrolidin-1-yl)propan-1-one
N-(1-{[(furan-2-ylmethyl)carbamoyl]methyl}-1H-pyrazol-4-yl)-2-(phenylsulfanyl)acetamide
2-[1-(6-aminopyridin-2-yl)-1H-pyrazol-3-yl]-4-chlorophenol
4-(2-methoxy-5-methylphenyl)-3-[(propan-2-yloxy)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(4-tert-butylphenoxymethyl)-5-(4,4-difluoropiperidine-1-carbonyl)pyrimidin-4-ol
3-phenyl-N-(1-{1-[(2,3,6-trifluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
(1S,5R)-6-methyl-3-[(3-methyl-1-benzofuran-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
ethyl 5-[(3-ethoxy-4-methoxyphenyl)methyl]-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-(4-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
1-(2H-1,3-benzodioxole-5-carbonyl)-3-[4-(3-chlorophenyl)-1H-pyrazol-5-yl]piperidine
N-[(2R,3R)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pentanamide
5-ethyl-5-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
[(3R,4R)-1-[6-(methoxymethyl)pyrimidin-4-yl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
3-(1-{5-[(diethylamino)methyl]-2-methylfuran-3-carbonyl}piperidin-3-yl)benzoic acid
6-(2,3-dihydro-1-benzofuran-2-carbonyl)-N-[4-(methylsulfanyl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
4-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-6-methoxypyrimidin-2-amine
N-methyl-3-(pyridin-4-yl)-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]propanamide
2-{4-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-{[(2,4-dimethylphenyl)carbamoyl]carbonyl}piperazin-1-yl)-N-ethylacetamide
(2S,4S)-4-{[(2,5-difluorophenyl)methyl]amino}-1-(2,3-dihydro-1H-inden-2-yl)-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
N-(2-{7-[(2,4-dimethoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-fluorobenzamide