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3-({5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)propan-1-ol
1-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(morpholin-4-yl)ethan-1-one
N-methyl-N-{1-[1-(4-methylbenzoyl)piperidin-4-yl]-2-(2-methylphenyl)ethyl}-2-(1H-pyrazol-1-yl)acetamide
methyl (2S,4R)-4-(dimethylamino)-1-[(2-methyl-1H-imidazol-4-yl)methyl]pyrrolidine-2-carboxylate
6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
(1R,5S,6S)-6-({2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}methyl)-3-azabicyclo[3.1.0]hexane
1-(azepan-1-yl)-3-[3-(1,4-oxazepan-4-ylmethyl)phenoxy]propan-2-ol
3-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-(3-methylpiperidin-1-yl)propan-1-one
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propan-1-one
6-cyclopentyl-N-[(4,6-dimethylpyridin-2-yl)methyl]-N,1-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(4-chlorophenyl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-phenylpropanamide
{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(thiophen-3-ylmethyl)amine
6-[(3-fluorophenyl)methoxy]-4-[(4-methyl-1H-imidazol-5-yl)methyl]-1-(2-methylpropyl)-1,4-diazepan-2-one
2-(1-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)-1,3-benzoxazole
3-hydroxy-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}pyridine-2-carboxamide
(3aR,6aR)-2-(2-cyclopentylacetyl)-5-(1H-imidazol-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(2-fluorophenoxymethyl)piperidine
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-3-(3-chlorophenyl)propan-1-one
N-[(2S,4R,6R)-2-(3,5-dimethoxyphenyl)-6-(4-fluorophenyl)oxan-4-yl]acetamide
ethyl 4-[(4-methoxyphenyl)methyl]-1-(oxolane-3-carbonyl)piperidine-4-carboxylate
1-[4-(piperidine-1-sulfonyl)-1,4-diazepan-1-yl]-2-(thiophen-2-yl)ethan-1-one
1-[1-(2-ethoxyacetyl)piperidin-3-yl]-3-phenylpropan-1-one
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]({[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
1-methyl-5-[4-(3-methylpyridin-2-yl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
8-(5-methoxy-1-methyl-1H-indole-2-carbonyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
8-[(4-oxo-4H-chromen-3-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-{1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1H-imidazol-2-yl}benzoic acid
N-cyclopropyl-3-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]oxy}-4-methoxybenzamide
[(4-fluorophenyl)methyl](methyl){[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-9-oxo-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide
5-chloro-N-(1-methoxypropan-2-yl)-15-methyl-13-oxo-9-(thiophen-3-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaene-12-carboxamide
methyl 3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(naphthalen-1-ylmethyl)piperidin-3-yl]propanoate
4-(2-aminopyridine-4-carbonyl)-1-(2-phenylphenyl)piperazin-2-one
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
3-(2-chlorophenyl)-4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}-5-methyl-1,2-oxazole
methyl(pyridin-3-ylmethyl)[2-(2,4,6-trifluorophenyl)ethyl]amine
3-acetamido-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]propanamide
1-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(pyridin-2-ylsulfanyl)ethan-1-one
8-(1-aminocyclopropanecarbonyl)-3-{3-[methyl(2-methylpropyl)amino]propyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[3-(5-methylfuran-2-yl)-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]morpholine
2-methoxy-N-(2-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}phenyl)acetamide
8-[(3R)-3-hydroxy-3-phenylpropyl]-8-azaspiro[4.5]decane-7,9-dione
4-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]benzamide
N-ethyl-2-methyl-3-[({[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}carbamoyl)amino]benzamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1-(3-methoxybenzoyl)piperidine
1-{4-[3-(morpholin-4-yl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
2-{1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}-N-(pyridin-2-ylmethyl)acetamide
2-methyl-N-(1-{7-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)propanamide
4-methyl-5-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2-(propan-2-yl)pyrimidine
4-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-2-(pyridin-3-yl)quinoline