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5-tert-butyl-N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]-1,3,4-oxadiazol-2-amine
{3-[(4-fluorophenyl)methyl]-1-[(4-methoxy-3-methylphenyl)methyl]piperidin-3-yl}methanol
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-2-(pyrrolidin-1-ylmethyl)piperidine
N-[(2R,3R)-1'-[3-(dimethylamino)benzoyl]-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
N-{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-N-(prop-2-yn-1-yl)cyclohexanamine
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4-(pyrrolidine-1-sulfonyl)-1,4-diazepane
N-(oxolan-2-ylmethyl)-3-{1-[3-(pyridin-3-yl)propanoyl]piperidin-4-yl}propanamide
(3-{2-[1-(3,6-dimethylpyrazin-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
9-[2-(propan-2-yloxy)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{1-azabicyclo[2.2.2]octan-3-yl}-8-fluoro-4-oxo-1,4-dihydroquinoline-3-carboxamide
5-(1H-indol-1-ylmethyl)-N-[2-(2-oxopiperidin-1-yl)ethyl]-1H-pyrazole-3-carboxamide
4-{[(4-methylphenyl)methyl]amino}-N-[(5-methylpyrazin-2-yl)methyl]benzamide
N-({2-[2-(2-cyclopentylacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-3,4-dimethylbenzamide
4-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,N,6-trimethylpyrimidin-2-amine
N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
2-[2-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)ethyl]-1,2,3,4-tetrahydrophthalazine-1,4-dione
3-methoxy-1-[(5-phenylthiophen-2-yl)methyl]pyrrolidine
4-fluoro-3-methoxy-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]benzamide
1-(4-methylpiperidin-1-yl)-3-[(thiolan-3-yl)amino]propan-1-one
8-methoxy-2-methyl-4-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(2-{imidazo[1,2-a]pyrimidin-2-yl}ethyl)amine
1-(1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-4-yl)-4-ethylpiperazine
N1-(4-methylpyridin-2-yl)-N2-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}ethane-1,2-diamine
N-[(3R,4R)-1-[(4-ethylphenyl)methyl]-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
3-[(3S,4R)-1-benzyl-4-(4-methylpiperazin-1-yl)piperidin-3-yl]-N-[2-(3,4-dimethoxyphenyl)ethyl]propanamide
(2S,4R)-4-amino-N,N-diethyl-1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)pyrrolidine-2-carboxamide
3-{[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]sulfamoyl}-N-(1,2-oxazol-3-ylmethyl)benzamide
1-(2-methylpropyl)-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
2-[5-(5,8-dimethoxy-4-methylquinolin-2-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
2-{2-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-2-oxoethyl}-4-methyl-1,2-dihydrophthalazin-1-one
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
N-[(1-cyclohexylpiperidin-3-yl)methyl]-2,3-dimethoxybenzamide
N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-2,2,3,3-tetramethylcyclopropane-1-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(diethylamino)methyl]phenoxy]-N-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]acetamide
[(3-{[1-(2,2-dimethyloxane-4-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](furan-3-ylmethyl)methylamine
7-[2-(2-ethoxyethoxy)benzoyl]-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-({1-[2-(1H-imidazol-4-yl)acetyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-4-hydroxy-2-methylpyrimidine-5-carboxamide
N-[3-(4-{[2-(dimethyl-1H-1,2,4-triazol-1-yl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-5-methylthiophene-2-carboxamide
N-(butan-2-yl)-7-acetamido-1-ethyl-2-(2-fluorophenyl)-1H-1,3-benzodiazole-5-carboxamide
(3R,4R)-1-[(4-chlorophenyl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
6,7-dimethoxy-2-(morpholin-4-ylmethyl)quinazolin-4-amine
2-oxo-8-{6-[(propan-2-yl)amino]pyrimidin-4-yl}-1,8-diazaspiro[4.5]decane-4-carboxylic acid
8-{imidazo[1,2-a]pyridine-3-carbonyl}-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-{[(2-fluorophenyl)methyl](methyl)amino}ethan-1-one
7-chloro-3,5-dimethyl-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1-benzofuran-2-carboxamide
4-benzyl-1-[(2,3-difluorophenyl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 5-{4-[2-(cyclopropylcarbamoyl)ethyl]piperidin-1-yl}-5-oxopentanoate
(2S,4R)-4-amino-N-methyl-1-[4-(1H-pyrrol-1-yl)benzoyl]pyrrolidine-2-carboxamide