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1-(4-chloro-2-fluorobenzoyl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
2-[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]-4-methyl-1H-1,3-benzodiazole
1-{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}-4-(methoxymethyl)piperidine
8-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
(3S,4S)-1-(2-ethoxypyridine-3-carbonyl)-4-propylpyrrolidine-3-carboxylic acid
2-(2-methoxyphenyl)-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
3-ethyl-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-4-methyl-1H-pyrazole-5-carboxamide
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(3-methylbut-2-en-1-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
8-(2H-1,3-benzodioxol-4-ylmethyl)-1-[(2-fluorophenyl)methoxy]-1,8-diazaspiro[4.5]decan-2-one
(3S,5R)-1-benzyl-N3-[(3,5-dimethylphenyl)methyl]-N5-(4-fluorophenyl)piperidine-3,5-dicarboxamide
3-[methyl({5-methylpyrazolo[1,5-a]pyrimidin-7-yl})amino]-1-phenylpropan-1-ol
4-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridin-6-yl]-6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaene
N-{[5-(2-chlorophenyl)-1,2-oxazol-3-yl]methyl}-1-(methoxymethyl)cyclobutane-1-carboxamide
1-[3-(furan-2-yl)benzoyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
1-{[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}-4-(propan-2-yl)piperazine
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
methyl (2S)-2-(3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamido)-3-phenylpropanoate
N-{1-[4-(1H-pyrazol-4-yl)butanoyl]piperidin-4-yl}benzamide
1-[(2R)-2-aminopropanoyl]-N-[3-(3-chlorophenyl)phenyl]piperidine-4-carboxamide
N-(3-{3,9-diazaspiro[5.6]dodecan-9-yl}-3-oxopropyl)-N-methylmethanesulfonamide
N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
1-[7-(cyclohexylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-4-methylpentane-1,2-dione
6-{3-[(4-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}-6-azabicyclo[3.2.1]octane
4-{[3-(furan-2-yl)propyl]sulfamoyl}-N-[(3S)-pyrrolidin-3-yl]benzamide
1-[(2S,6S)-6-(hydroxymethyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}pyridine-2-carboxamide
N-[3-(1H-indol-1-yl)propyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
1-{1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(pyridin-2-yl)piperazine
5-(cyclohex-3-ene-1-carbonyl)-3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-{[4-(3-chlorophenyl)-5-({[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl](methyl)amino}methyl)-4H-1,2,4-triazol-3-yl]sulfanyl}propan-1-ol
N-[(2-aminopyrimidin-5-yl)methyl]-N,2,6-trimethylquinoline-4-carboxamide
1'-{[3-methoxy-4-(propan-2-yloxy)phenyl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-{4-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]phenyl}morpholine
N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-3-phenyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-(2-methoxyphenyl)propanamide
(1-{[5-(oxan-2-yl)thiophen-2-yl]methyl}-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)methanol
3-(3-chloro-1,2-oxazol-5-yl)-N-[(2,3-dimethyl-1H-indol-5-yl)methyl]propanamide
5-{[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]methyl}isoquinoline
[3-(3-methylbut-2-en-1-yl)-1-(oxane-4-carbonyl)piperidin-3-yl]methanol
N-(dimethyl-1,2-oxazol-4-yl)-2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carboxamide
(2R,3R,6R)-3-(2-methoxyphenyl)-5-(3-methylbenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-[(1-acetylpiperidin-4-yl)oxy]-N-benzyl-5-methoxy-N-methylbenzamide
5-[4-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)phenyl]-1H-pyrazole
1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
2-[3-(4-fluorophenyl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-indazol-3-yl)acetamide
6-{[(1S,2S)-2-hydroxycyclohexyl]amino}-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}piperidin-3-amine
1-[2-(3-chlorophenyl)ethyl]-4-[(4-methylpyrimidin-2-yl)amino]pyrrolidin-2-one
2-{2-[3-benzyl-3-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindole-1,3-dione
1-cyclohexyl-N-[2-(1H-pyrrol-1-yl)ethyl]piperidine-4-carboxamide