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8-[4-methyl-6-(methylamino)pyrimidin-2-yl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-fluoro-N-[2-(1,2-oxazol-3-ylformamido)ethyl]benzamide
1-[3-(dimethylamino)benzoyl]-N-(4-methoxyphenyl)piperidin-3-amine
1-cyclohexyl-4-[3-(2-oxopyrrolidin-1-yl)benzoyl]-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
1-ethyl-3-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
5-acetyl-N-{[3-methyl-7-(5-methyl-1H-pyrazole-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-3-carboxamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-[(cyclopropylmethyl)sulfanyl]acetamide
(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-2-[2-(4H-1,2,4-triazol-4-yl)ethyl]-decahydroisoquinoline
1-cyclopentyl-N-(3-methylbutyl)-4-oxo-5-(4-phenylpiperazine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-N,N-dimethylpyrrolidin-3-amine
4-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
2-[2-(dimethylamino)ethyl]-9-(2,6-dimethylpyrimidine-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
6-methyl-N-[1-(oxolan-2-ylmethyl)piperidin-4-yl]imidazo[1,2-a]pyridine-2-carboxamide
1-(1H-pyrazol-3-ylmethyl)-3-[3-(trifluoromethyl)benzoyl]piperidine
N-[(3R,4R)-1-[(8-fluoroquinolin-2-yl)methyl]-3-hydroxypiperidin-4-yl]pyridine-4-carboxamide
4-({4-methyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}methyl)morpholine
8-methoxy-N-[3-(morpholin-4-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-amine
3-(3-methoxyphenyl)-N-{[8-(thiophene-2-sulfonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}propanamide
(4aS,8aR)-1-butyl-6-[2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
4-{[2-(pyridin-4-yl)phenyl]methyl}morpholine
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-(3-phenylpropyl)-1H-pyrazole-3-carboxamide
(2S)-2-acetamido-N-[(4-fluorophenyl)methyl]-N-(prop-2-en-1-yl)propanamide
methyl 5-[(4-hydroxy-4-methylpentan-2-yl)amino]-1-(2-methylpropyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
[5-({[(2-methoxyphenyl)methyl](pyridin-3-ylmethyl)amino}methyl)furan-2-yl]methanol
N-methyl-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-3-(4H-1,2,4-triazol-4-yl)benzamide
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
5-{[(1R,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-2,1,3-benzothiadiazole
1-methyl-4-[1-(1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidin-4-yl)ethyl]piperazine
ethyl 1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-4-(3-phenylpropyl)piperidine-4-carboxylate
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)acetamide
methyl 8-[(2E)-2-methylbut-2-en-1-yl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
2-{[2-cyclopropyl-7-(4-methyl-1H-imidazole-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethan-1-ol
1-ethyl-5-{1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-imidazol-2-yl}-1H-1,2,4-triazole
1-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
8-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
8-[(6-carboxypyridin-2-yl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-[(1S,5R)-6-benzyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N-(thiophen-2-ylmethyl)acetamide
3-{[(2-methoxyethyl)(methyl)amino]methyl}-N,8-dimethyl-N-(2-phenylethyl)imidazo[1,2-a]pyridine-2-carboxamide
3-hydroxy-3-({[(2-hydroxypyridin-3-yl)methyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(3-phenylpropyl)acetamide
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(2,4-difluorophenoxy)acetamide
(1S,4S)-2-[5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-2-azabicyclo[2.2.1]heptane
ethyl 5-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(1R,4S)-N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]heptane-4-carboxamide
5-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
2-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-fluoropyridine
1-(6-cyclopropylpyrimidin-4-yl)-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
3-butyl-1-methyl-4-[4-(5-methylfuran-2-yl)benzoyl]piperazin-2-one
3-[2-(4-hydroxy-2-methoxyphenyl)-1H-imidazol-1-yl]piperidin-2-one
N-(1-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide