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4-[5-(6-methylpyridine-3-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
1-[(3-chlorophenyl)methyl]-3-(ethoxymethyl)-5-(oxolan-3-yl)-1H-1,2,4-triazole
2-{[(2-methoxyethyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amino]methyl}benzoic acid
1-[(4-methyl-1,4-oxazepan-6-yl)methyl]-3-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}urea
1-(4-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}piperidin-1-yl)ethan-1-one
3-cyclopropyl-5-[1-(2,5-difluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1H-pyrazole
2-acetyl-7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-[cyclohexyl(methyl)amino]-3-[4-({[2-(furan-2-yl)ethyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
3-{[2-(furan-2-yl)-7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl]methyl}-1λ6-thiolane-1,1-dione
1-methyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazole
N,N-diethyl-2-({4-[2-(3-fluorophenyl)acetyl]-1-[(4-methoxyphenyl)methyl]-2-oxo-1,4-diazepan-6-yl}oxy)acetamide
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{2-[4-(trifluoromethyl)phenyl]ethyl}propanamide
2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-(2-methylbutyl)acetamide
6-(aminomethyl)-2-methyl-N-[(1R,2S)-2-phenylcyclopropyl]pyrimidin-4-amine
[3-(2-methoxyethyl)-1-(thiophene-3-carbonyl)piperidin-3-yl]methanol
1-(2,3-dihydro-1H-inden-2-yl)-N-({4-[2-(pyrimidin-5-yl)ethynyl]phenyl}methyl)piperidin-3-amine
2-(dimethylamino)-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-(4-fluorophenyl)-N-methylacetamide
2-chloro-N-[2-(oxane-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]benzamide
4-[1-cyclohexyl-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-1-(oxolane-2-carbonyl)piperidine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-7-fluoro-2-oxo-1,2-dihydroquinoline-4-carboxamide
2,5,7-trimethyl-N-({8-[(2-methylphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)quinoline-4-carboxamide
N-[2-(1H-imidazol-4-yl)ethyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-4-oxo-3,4-dihydrophthalazine-1-carboxamide
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-[(2-methylpyrimidin-5-yl)methyl]piperidine-4-carboxylic acid
N-{4-[4-(4-phenylazepan-1-yl)piperidin-1-yl]phenyl}pyrazine-2-carboxamide
3-(3-methoxyphenyl)-5-{1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1H-pyrazole
3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-{4-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-5-(thiomorpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole
4-[6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-3,3-dimethylpiperazin-2-one
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
(3S,9aR)-8-[(3-fluoro-4-methylphenyl)methyl]-3-(1H-imidazol-4-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-{[1-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)piperidin-4-yl]methyl}morpholine
1-(2-methoxyethyl)-N-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
(3aR,6aR)-2-[1-(methoxymethyl)cyclobutanecarbonyl]-5-(pyridin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-chloro-2-[3-(2-methoxyphenoxy)azetidin-1-yl]quinoline
8-fluoro-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}quinoline-2-carboxamide
N-benzyl-1-(4,7-dimethylquinazolin-2-yl)piperidine-4-carboxamide
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(2-methoxyphenyl)acetamide
2-(1-methyl-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl)ethan-1-ol
2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-4-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1,3-oxazole
N-{[3-methyl-7-(1-phenylcyclopropanecarbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(piperidin-1-yl)acetamide
N-benzyl-N-methyl-3-({[3-(pyridin-3-yloxy)propyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
N-cyclopropyl-5-(1,2,3,6-tetrahydropyridin-4-yl)thiophene-2-carboxamide
(2R,6R)-4-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4-({[(5-methylthiophen-2-yl)methyl]carbamoyl}amino)-N-(oxolan-2-ylmethyl)benzamide
1-(1-phenylcyclohexanecarbonyl)-4-(pyridin-3-ylmethyl)-1,4-diazepan-5-one
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
(2R,6R)-4-(1H-imidazol-2-ylmethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-(dimethyl-1,2-oxazol-4-yl)urea
4-{1-methyl-3-[(E)-2-[4-(trifluoromethyl)phenyl]ethenyl]-1H-1,2,4-triazol-5-yl}morpholine