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1-(4-{2-[2-(3-methoxyphenyl)ethyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)-2-(thiophen-3-yl)ethan-1-one
3-(1H-imidazol-4-yl)-2-{[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}propanoic acid
2,6-dimethoxy-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pyridine-3-carboxamide
9-(4-methyl-1,3-thiazole-5-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{6-[4-(piperidin-1-ylmethyl)piperidin-1-yl]pyridin-2-yl}ethan-1-ol
1-cyclopentyl-4-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carbonyl}-1,4-diazepane
(4aS,8aR)-1-butyl-6-[1-(1H-imidazol-1-ylmethyl)cyclopropanecarbonyl]-decahydro-1,6-naphthyridin-2-one
2-(4-chlorophenyl)-2-[3-(trimethyl-1H-pyrazol-4-yl)propanamido]acetic acid
2-{[(2-chlorophenyl)methyl]sulfanyl}-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
N-[(2R,3R)-2-methoxy-1'-(naphthalen-2-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
1-(1-benzylpiperidin-4-yl)-N-methyl-N-(3-methylbutyl)piperidine-3-carboxamide
4-[(4-fluorophenyl)methyl]-1-(2-methylbenzoyl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
methyl 2-[1-({4-[ethyl(2-methylprop-2-en-1-yl)amino]quinazolin-2-yl}methyl)-3-oxopiperazin-2-yl]acetate
1-(azepan-1-yl)-3-{3-[({[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}amino)methyl]phenoxy}propan-2-ol
methyl 2-[4-(5-{[(2-methoxyphenyl)carbamoyl]amino}-1H-pyrazol-1-yl)piperidin-1-yl]acetate
2-{[1-(cyclohexylmethyl)piperidin-4-yl]oxy}-4-methoxy-N-(2-methoxyethyl)benzamide
2-(2-methoxyphenyl)-1-[4-(4H-1,2,4-triazol-3-ylmethyl)piperazin-1-yl]ethan-1-one
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]({[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
N-(cyclohex-1-en-1-ylmethyl)-2-(1-ethylpiperidin-4-yl)acetamide
4-[({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)carbamoyl]pyridin-1-ium-1-olate
(5-{[(butan-2-yl)(pyridin-4-ylmethyl)amino]methyl}furan-2-yl)methanol
4-{3-[3-(morpholin-4-yl)piperidine-1-carbonyl]phenyl}morpholine
1,1-dioxo-N-[3-(2-oxo-1,2-dihydropyridin-1-yl)propyl]-3,4-dihydro-2H-1λ6,2-benzothiazine-3-carboxamide
2-methyl-N-(1-{7-[(3-methylthiophen-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)propanamide
3-{5-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]-1H-1,3-benzodiazol-1-yl}propan-1-ol
2,3,4-trimethoxy-N-{[5-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
ethyl 4-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperazine-1-carboxylate
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-[1-(thiophen-2-yl)propyl]piperidine-4-carboxamide
5-{1-[(3,4-dimethylphenyl)methyl]piperidin-4-yl}-5-[(3-methoxyphenyl)methyl]-3-methylimidazolidine-2,4-dione
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-(1H-imidazol-1-yl)propanamide
N-(2-hydroxyethyl)-2,6-dimethoxy-N-[(2E)-3-phenylprop-2-en-1-yl]pyridine-3-carboxamide
5-methanesulfonyl-4-(piperidin-3-yl)-N-[2-(pyrrolidin-1-yl)ethyl]pyrimidin-2-amine
8-[4-(furan-2-yl)benzoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-{[7-(3-chloro-4-fluorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(thiophen-2-yl)acetamide
(3R,4S)-4-phenyl-1-(pyridazine-3-carbonyl)pyrrolidin-3-amine
3-(2-chlorophenyl)-3-{2-[4-(1-hydroxypropyl)piperidin-1-yl]-2-oxoethyl}-1-(2-methoxyethyl)pyrrolidine-2,5-dione
4-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-3-propylmorpholine
1-{1-[1-(2-phenylethyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]ethyl}pyrrolidin-2-one
2-(pyridin-2-yl)-5-[4-(pyrimidin-2-yloxy)piperidine-1-carbonyl]pyrimidin-4-ol
1-[(1R)-2-hydroxy-1-phenylethyl]-3-[3-(4-methylpiperidine-1-carbonyl)phenyl]urea
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-(1H-pyrazol-4-yl)butanamide
N-[4-(4-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}piperidin-1-yl)phenyl]cyclopentanecarboxamide
2-(oxane-4-carbonyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]pyrrolidin-3-yl]urea
N2-[4-(1,3-benzoxazol-2-yl)phenyl]-N1-ethylpyrrolidine-1,2-dicarboxamide
3-{4-[2-(1,2-oxazolidine-2-carbonyl)phenoxy]piperidine-1-carbonyl}pyridine
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-[(3-methylpyridin-2-yl)methyl]piperazine
2-cyclopropyl-N-(2,5-difluorophenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(pyridin-4-ylsulfanyl)ethan-1-one