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2-[(3-{[2-(cyclohexylcarbamoyl)ethyl]carbamoyl}phenyl)amino]acetic acid
1-methyl-3-[3-(2-methylphenyl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1H-indazole
N-[2-(1H-imidazol-4-yl)ethyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
6-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}pyridine-2-carbonitrile
8-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-(1-methylpiperidine-3-carbonyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
5-(2,6-difluorophenoxymethyl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,2-oxazole-3-carboxamide
3-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-chloro-2-methylphenyl)urea
2-(2-methoxyphenyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)acetamide
2-ethyl-4-methyl-5-{[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-imidazole
N-cyclohexyl-N-(2-hydroxyethyl)-2-methyl-1-benzofuran-5-carboxamide
3-{4-[(4-ethyl-3-oxopiperazin-1-yl)methyl]-1H-pyrazol-1-yl}propanoic acid
(2R,6S)-4-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,6-dimethylmorpholine
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-8-fluoroquinoline-2-carboxamide
methyl 2-[3-(1-acetamido-3-methylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]benzoate
1-(4-cyclopentylpiperazin-1-yl)-3-(2-hydroxyphenyl)-3-(3-hydroxyphenyl)propan-1-one
1-[2-(2-chlorophenyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl]-4-(methoxymethyl)piperidine
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-[(3-methoxyphenyl)methyl]-N-methylpropanamide
N-[1-(2,2-dimethylpent-4-en-1-yl)piperidin-4-yl]methanesulfonamide
2-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-phenylacetamide
N-{[7-fluoro-5-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-4-methyl-1H-imidazole-5-carboxamide
1-(2,2-dimethylpropyl)-3-hydroxy-3-({[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]amino}methyl)piperidin-2-one
3-(1-ethyl-1H-imidazol-2-yl)-1-(2-propoxybenzoyl)piperidine
methyl 1-(naphthalen-2-ylmethoxy)-2-oxo-8-(pyridin-4-ylmethyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
5-benzamido-1-cyclopentyl-N-(2-methoxyethyl)-N-methyl-1H-1,3-benzodiazole-7-carboxamide
methyl 2-({2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}methyl)-1,3-oxazole-4-carboxylate
3-(3-hydroxyquinoxalin-2-yl)-N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)propanamide
4,5-dimethyl-6-[4-(piperidine-1-sulfonyl)-1,4-diazepan-1-yl]pyrimidin-2-amine
methyl 2-{8-[(3,4-dimethoxyphenyl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl](methyl)[3-(pyrrolidin-1-yl)propyl]amine
8-fluoro-N-[1-(morpholine-4-carbonyl)piperidin-4-yl]quinoline-2-carboxamide
3-[(3R,4S)-1-(1-methyl-1H-indole-4-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
(1S,5R)-N-(furan-2-ylmethyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
9-methoxy-3-[(3-methoxyphenyl)methyl]-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-fluoro-4-methoxy-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]benzamide
4-methyl-6-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}-2-(pyridin-3-yl)pyrimidine
N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-2-(trifluoromethyl)benzene-1-sulfonamide
5-[1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-5-(3-phenylpropyl)imidazolidine-2,4-dione
5-{2-[4-(3-methylpyridin-2-yl)piperazin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-(3-carbamoyl-4-fluorophenyl)-4-(pyridin-2-ylmethoxy)piperidine-1-carboxamide
1-[(2-chlorophenyl)methyl]-N-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1H-1,2,3-triazole-4-carboxamide
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-(2,3-dimethylphenyl)-N'-ethyl-N'-{[3-(prop-2-en-1-yloxy)phenyl]methyl}propanediamide
1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-4-(2-methoxyphenyl)-2-methylpiperazine
4-cyclopropyl-6-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]pyrimidine
3-{1-[(2-chloro-6-fluorophenyl)methyl]piperidin-4-yl}-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
2-{4-phenyl-5-[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]-1H-imidazol-1-yl}ethan-1-ol
5-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]-N,N,4-trimethylpyrimidin-2-amine