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(4aR,7aS)-1-(2-hydroxyethyl)-4-(2,4,5-trimethylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(3-fluorophenyl)-6-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-1-[2-(piperidin-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(methylamino)-1,3-thiazole-4-carboxamide
1-[(2-fluorophenyl)methoxy]-8-{2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]acetyl}-1,8-diazaspiro[4.5]decan-2-one
3-methoxy-1-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]propan-1-one
1-(1H-1,2,3-benzotriazol-5-yl)-3-ethyl-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]urea
1-{1-[2-(1H-indol-3-yl)acetyl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
2-methyl-6-{4-[1-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-ol
(4aR,7aS)-1-(2-methoxyethyl)-4-(2-phenoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-[2-(methylsulfanyl)ethyl]acetamide
ethyl 5-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(2R,4S)-4-hydroxy-1-{4-[(2-methylprop-2-en-1-yl)oxy]benzoyl}piperidine-2-carboxylic acid
2-[1-cyclohexyl-3-(2-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-[(3,4-dimethoxyphenyl)methyl]-N-methylacetamide
N-{3-[3-(3-chloro-2-methylphenyl)-1,2,4-oxadiazol-5-yl]propyl}acetamide
3-(3-hydroxy-3-methylbutyl)-N-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)benzamide
methyl 8-[(2-fluorophenyl)methyl]-2-oxo-1-propoxy-1,8-diazaspiro[4.5]decane-4-carboxylate
2-cyclopropyl-N-[3-(methylsulfanyl)propyl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]pent-4-enamide
N-(1H-imidazol-2-ylmethyl)-N,3-dimethyl-5-propyl-1-benzofuran-2-carboxamide
5-fluoro-2-[1-(5-phenyl-1,2,4-triazin-3-yl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
4-methyl-5-[3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)propyl]-1,3-thiazole
(4aR,8aS)-6-(9H-fluoren-2-ylmethyl)-1-[(4-fluorophenyl)methyl]-decahydro-1,6-naphthyridin-2-one
2-cyclohexyl-1-[3-(3-methoxybenzoyl)piperidin-1-yl]ethan-1-one
N-[4-(2,2-dimethylpropanamido)-3-methylphenyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
3-[(3R,4S)-3-amino-4-phenylpyrrolidine-1-carbonyl]-1,6-dimethyl-1,4-dihydroquinolin-4-one
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(1,3-thiazol-2-ylmethyl)pyridin-2-amine
4-[(3-chloro-2-fluorophenyl)methyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
1-(butan-2-yl)-N3-cyclooctyl-N5-ethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
methyl 2-{4-phenyl-5-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}acetate
1-{4-[(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)methyl]thiophen-2-yl}ethan-1-one
5-fluoro-2-[4-(1H-pyrazol-1-yl)phenyl]phenol
{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}(2,3-dihydro-1-benzofuran-2-ylmethyl)methylamine
1-cyclopropyl-N-methyl-6-oxo-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidine-3-carboxamide
3,3-dimethyl-1-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]butan-1-one
2-{1-[6-(4-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidin-2-yl}ethan-1-ol
7-[(2,3-dimethoxyphenyl)methyl]-2-ethyl-2,7-diazaspiro[4.5]decane
2-[4-fluoro-3-(trifluoromethyl)phenyl]-N-methylpyrimidin-4-amine
5-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine-2-carbonitrile
N-[(5-chloro-2-propoxyphenyl)methyl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propanamide
(4aR,7aS)-1-(2-methoxyethyl)-4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{5-[1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
1-[(2-methoxyphenyl)methyl]-N-[(2-methyl-1H-indol-5-yl)methyl]-6-oxopiperidine-3-carboxamide
4-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}-1-methylpiperazine-2-carboxylic acid
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-2-propyl-1,3-thiazole-4-carboxamide
4-[1,3-dimethyl-5-(morpholin-4-yl)-1H-pyrazol-4-yl]-7-hydroxy-6-methyl-1,2,3,4-tetrahydroquinolin-2-one
1-(3-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-3-oxopropyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-(1H-imidazol-2-ylmethyl)benzamide
3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[2-(piperidin-1-yl)ethyl]propanamide
[(3S,5R)-1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol