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3-{[3-(morpholin-4-yl)azetidin-1-yl]methyl}benzoic acid
1-[3-(4-fluorophenoxy)propyl]-4-(1-methylpiperidine-4-carbonyl)piperazine
2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-4-(3,3,3-trifluoropropyl)pyrimidine
4-{6-[(dimethylamino)methyl]-1,4-oxazepane-4-carbonyl}benzene-1-sulfonamide
N,N,4-trimethyl-3-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-N-[2-(4-phenylpyrimidin-2-yl)ethyl]acetamide
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[1-(naphthalen-1-yl)ethyl]propanamide
2-[3-cyclopropyl-5-(3-methyl-1,2-oxazol-5-yl)-1H-1,2,4-triazol-1-yl]pyridine
1-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-3-(1H-imidazol-2-yl)piperidine
methyl 2-({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)-1,3-oxazole-4-carboxylate
2-cyclohexyl-7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-(but-2-yn-1-yl)-5-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
4-{[1-(furan-3-ylmethyl)piperidin-4-yl]oxy}-N-(pyridin-4-ylmethyl)benzamide
2-ethoxy-5-methyl-N-[(1-methylpiperidin-3-yl)methyl]benzene-1-sulfonamide
8-(5-ethyl-1,3-oxazole-4-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(2-methoxyethyl)-5-({4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}methyl)pyrimidine
6-methyl-2-(1-{[3-(3-methylbutyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-yl)-1H-1,3-benzodiazole
7-(2,3,4,9-tetrahydro-1H-carbazole-8-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
N-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-3-(1-methylpiperidin-2-yl)propanamide
2-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-6-phenylpyridine-3-carboxylic acid
(3E)-N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}hex-3-enamide
3-methoxy-N-methyl-4-[(1-methylpiperidin-4-yl)oxy]-N-[1-(1,2-oxazol-3-yl)ethyl]benzamide
2-methoxy-5-({methyl[(1,2,2-trimethylpyrrolidin-3-yl)methyl]amino}methyl)benzoic acid
1-(1,3-dioxo-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindol-4-yl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)piperidine-4-carboxamide
1-(carbamoylmethyl)-N-[2-(4-chlorophenyl)-2-hydroxyethyl]piperidine-4-carboxamide
1-{[2-fluoro-3-(2-methoxy-5-methylphenoxy)phenyl]methyl}pyrrolidine
1-[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-hydroxyethan-1-one
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
5-{[benzyl(3-hydroxy-2-methylpropyl)amino]methyl}-2-methoxybenzoic acid
5-({5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}amino)pentan-1-ol
3-{5-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-7-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
(3S)-3-ethyl-4-{[5-(pyridin-2-yl)thiophen-2-yl]sulfonyl}morpholine
4-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridin-6-yl]-5-ethyl-6-methylpyrimidin-2-amine
{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})amine
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1-oxo-2-[2-(pyridin-4-yl)ethyl]-2,3-dihydro-1H-isoindole-5-carboxamide
1-{2-[3-(piperidin-1-yl)azetidine-1-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}ethan-1-one
1-(1,3-benzothiazole-6-carbonyl)-N-(pyridin-2-ylmethyl)piperazine-2-carboxamide
2,2-dimethyl-N-(1-{1-[2-(1H-pyrazol-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
3-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-oxoethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-2-one
N-{1-[1-(3-aminopropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-phenylmethanesulfonamide
1-[(3-methylthiophen-2-yl)methyl]-4-[2-(2-phenylethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
3-[2-(dimethylamino)ethyl]-5-{1-[(2E)-3-(4-methoxyphenyl)prop-2-enoyl]piperidin-4-yl}-5-(3-methylbutyl)imidazolidine-2,4-dione
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[(tert-butylcarbamoyl)methyl]pyrrolidine-3-carboxylic acid
2-ethyl-1-[6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidine
4-propyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)pyrimidine-5-carboxamide
N,2-dimethyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]thieno[2,3-d]pyrimidin-4-amine
4-(2-ethylpyridine-4-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(1s,4s)-4-[3-(3-methoxyphenoxymethyl)piperidine-1-carbonyl]cyclohexan-1-ol