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N-[2-(4-hydroxyphenyl)-2-oxoethyl]-1-methanesulfonyl-N-methylpyrrolidine-2-carboxamide
8-[(2-ethylpyrimidin-5-yl)methyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-{[(1s,4s)-4-aminocyclohexyl]methyl}pyrrolidine-3-carboxylic acid
5-[1-(2-cyclopropylacetyl)piperidin-4-yl]-5-propyl-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
2-[1-cyclopropyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-(2-methoxyethyl)-N-methylacetamide
1-benzyl-N3-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-amino-6-ethyl-4-(4-hydroxy-3,5-dimethoxyphenyl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile
1-{1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-[3-(trifluoromethyl)phenyl]piperazine
N-[2-(dimethylamino)ethyl]-5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-pyrazole-3-carboxamide
3-fluoro-N-({7-[(4-fluoro-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
N-[2-(azepan-1-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-(1-{7-[(4-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclopropanecarboxamide
1-amino-N-({1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}methyl)cyclopentane-1-carboxamide
N,1-dimethyl-N-{1-[1-(3-methylbutyl)piperidin-4-yl]-2-phenylethyl}-1H-pyrazole-3-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-6-[(4-oxo-4H-chromen-3-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
3-(2-methoxybenzoyl)-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidine
6-(aminomethyl)-2-(4-{[(2,3-dihydro-1-benzofuran-2-ylmethyl)(methyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
2-(adamantan-1-yl)-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4-[(3-methylpyridin-2-yl)methyl]piperazine
N-(2-{7-[(2-methoxynaphthalen-1-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
N-({7-[(2,4-dimethoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-phenylacetamide
3-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]-1,2-dihydroquinoxalin-2-one
(3R,5R)-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
methyl 6-{2-[(4-phenylbutanamido)methyl]-2,3-dihydro-1-benzofuran-7-yl}pyridine-3-carboxylate
4-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
(2H-1,3-benzodioxol-4-ylmethyl)(methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
N,2-dibenzyl-N-(2-hydroxyethyl)-1,3-benzoxazole-5-carboxamide
N-(pyridin-2-ylmethyl)-5-(1H-pyrrole-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
5-{1-[(8-methoxy-2H-chromen-3-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
5-cyclobutanecarbonyl-1'-(thiophen-2-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2,5-dimethyl-N-(3-{5-methyl-4-[(2-methylbutanamido)methyl]-1,3-oxazol-2-yl}phenyl)furan-3-carboxamide
N'-[(1-{[6-(trifluoromethyl)pyridin-3-yl]methyl}pyrrolidin-3-yl)methyl]ethanediamide
1-{1-[(2-chloro-6-fluorophenyl)methyl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
methyl 5-cyano-6-[4-(acetamidomethyl)piperidin-1-yl]-2-methylpyridine-3-carboxylate
4-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-cycloheptyl-N-[(5-methylpyrazin-2-yl)methyl]-6-oxopiperidine-3-carboxamide
3-methoxy-2-({3-[4-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
(4aS,8aS)-2-(2,3-difluorobenzoyl)-decahydro-2,7-naphthyridin-4a-ol
1-(6-methyl-1H-1,3-benzodiazol-7-yl)-3-[(1-propyl-1H-imidazol-2-yl)methyl]urea
3,5-dimethyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-1H-pyrazole-4-sulfonamide
benzyl 3-[2-(5-acetylthiophen-3-yl)acetamido]pyrrolidine-1-carboxylate
4-[(3-{2-[4-(2,6-dimethoxybenzoyl)piperazin-1-yl]ethoxy}phenyl)methyl]morpholine
methyl (2S,4S)-4-[(cyclohexylcarbamoyl)amino]-1-methylpyrrolidine-2-carboxylate
3-[(4-fluorophenyl)methyl]-5-[1-(1-methylcyclopropanecarbonyl)piperidin-4-yl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
N-(pentan-3-yl)-1-(thiophene-2-carbonyl)piperidin-3-amine
N-[2-(1H-imidazol-4-yl)ethyl]-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
5-(3,4-difluorophenoxymethyl)-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
1-[2-methoxy-5-(piperidin-1-ylmethyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
(3S,4R)-4-methyl-1-[3-(1,3-thiazole-2-carbonyl)pyridin-2-yl]piperidine-3,4-diol