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N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-5-methylthiophene-2-carboxamide
N6-cyclopentyl-N5-methyl-N5-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
[(6-methoxy-2H-chromen-3-yl)methyl](methyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
methyl (2S)-1-{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}pyrrolidine-2-carboxylate
N-(1H-indol-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[2-(oxan-2-yl)ethyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
1-[cyclopropyl(4-methylpyridin-2-yl)methyl]-3-(3-methylcinnolin-5-yl)urea
3-(but-2-yn-1-yl)-5-(3-phenylpropyl)-5-[1-(thiophene-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazine
6-fluoro-2-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
1-({2-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]phenyl}methyl)-1H-pyrazole
7-[4-methyl-7-(methylsulfanyl)quinolin-2-yl]-2,7-diazaspiro[4.4]nonane-1,3-dione
2-phenyl-7-(1-propyl-1H-pyrazole-5-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
methyl 2-({[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxylate
5-(2-{2-[4-(3-hydroxyphenyl)-1H-1,2,3-triazol-1-yl]ethyl}morpholin-4-yl)-2-methyl-2,3-dihydropyridazin-3-one
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-(3-cyclopropylpropanoyl)-decahydro-1,6-naphthyridin-2-one
[(1-cyclopentylpiperidin-4-yl)methyl][(3-fluorophenyl)methyl](oxolan-2-ylmethyl)amine
N-{[8-(pyridin-2-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-1H-indole-6-carboxamide
N-(1-propylcyclopropyl)-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
1-[2-(3-fluorophenyl)ethyl]-5-[4-(2-methoxyethoxy)piperidine-1-carbonyl]piperidin-2-one
N-{[3-methyl-7-(2,2,3,3-tetramethylcyclopropanecarbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(1-methyl-1H-1,2,3-triazol-4-yl)urea
N-(3,5-dimethylphenyl)-6-{2-[3-(trifluoromethyl)phenyl]acetyl}-6-azaspiro[2.5]octane-1-carboxamide
N-[(2-chlorophenyl)methyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-methyl-5-{4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
3-(4-chloro-1H-pyrazol-1-yl)-1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]propan-1-one
7-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[2-(2-oxopyrrolidin-1-yl)ethyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(2S)-2-{[3-ethoxy-4-(prop-2-en-1-yloxy)phenyl]formamido}pentanedioic acid
N-{4-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-4-oxobutan-2-yl}acetamide
4-chloro-N-{3-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}benzamide
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
2-[(4aR,7aS)-4-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
7-chloro-3-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}-3,4-dihydroquinazolin-4-one
3-butyl-4-(6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-methylpiperazin-2-one
6-methyl-1-{3-[2-(morpholin-4-ylmethyl)piperidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
2-methoxy-3-[3-(pyridin-2-yl)azetidine-1-carbonyl]pyridine
2-[3-(2-methoxyethyl)-5-[6-(methoxymethyl)pyridin-2-yl]-1H-1,2,4-triazol-1-yl]acetic acid
(1S,6R)-9-[(2-hydroxy-7-methoxyquinolin-3-yl)methyl]-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(furan-2-yl)-1H-pyrazole-4-carboxamide
(3S,9aR)-8-benzyl-3-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(1-{1-[3-(2-oxopyrrolidin-1-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
1-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}-3-(1,2-oxazolidin-2-yl)propan-1-one
3-{1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}-N-(2-chlorophenyl)propanamide
2-(2-hydroxyethyl)-8-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
4-(4-fluorophenyl)-3-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazole
2-cyclohexyl-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1,3-benzoxazole-6-carboxamide
1-(2-methylpyridin-4-yl)-4-[2-(methylsulfanyl)pyridine-3-carbonyl]-1,4-diazepane
(3aR,6aR)-2-(2-methoxyethyl)-5-{2-[4-(methylsulfanyl)phenyl]acetyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-4,6-dimethylpyridine-3-carbonitrile