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6-[2-(2-methylphenyl)acetyl]-N-(3-phenylpropyl)-6-azaspiro[2.5]octane-1-carboxamide
N-[(6-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
2-(1H-indol-3-yl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-[(2R,3R)-2-methoxy-1'-[2-(4-methylphenoxy)acetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
3-{5-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
3-{N-benzyl-1-[3-(5-methylfuran-2-yl)phenyl]formamido}propanamide
N-cyclopropyl-3-{1-[5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carbonyl]piperidin-4-yl}propanamide
N-{4-[4-(benzylamino)piperidin-1-yl]phenyl}cyclopentanecarboxamide
3-[(4-ethoxyphenyl)methyl]-9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-[(2-chlorophenyl)methyl]-N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N-(4-butylphenyl)-4-(4H-1,2,4-triazol-4-yl)piperidine-1-carboxamide
4-{5-[(4-{1-azabicyclo[2.2.2]octan-3-yl}piperazin-1-yl)methyl]thiophen-2-yl}-2-methylbut-3-yn-2-ol
4-(1-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}azetidin-3-yl)morpholine
6-(2-chlorophenyl)-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
5-[3-(3-acetylpiperidin-1-yl)-3-oxopropyl]-5-[(2-fluoro-4-methoxyphenyl)methyl]pyrrolidin-2-one
3-(4-methoxy-3,5-dimethylbenzoyl)-1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidine
{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)[(4-methyl-1,3-thiazol-2-yl)methyl]amine
4-[2-(2H-indazol-2-yl)acetyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
2-(5-acetylthiophen-3-yl)-1-[2-(3-methoxyphenyl)azetidin-1-yl]ethan-1-one
2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]acetamide
9-{[6-(dimethylamino)pyridin-3-yl]methyl}-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-3-(1H-1,2,4-triazol-1-yl)propanamide
(1R,7S)-N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-3-(4-fluorophenyl)-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
[1-({[6-(propan-2-yl)pyrimidin-4-yl]amino}methyl)cyclobutyl]methanol
3-[(cyclobutylamino)methyl]-1-(2-cyclohexylethyl)-3-hydroxypiperidin-2-one
2-[(3,4-dimethoxyphenyl)methyl]-N-(3-ethoxy-2-hydroxypropyl)-1,3-benzoxazole-6-carboxamide
methyl 2-(diethylsulfamoyl)-6-(2-phenoxypropanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-{1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}-5-(3-methylbutyl)imidazolidine-2,4-dione
2-(2,3-dihydro-1H-inden-1-yl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}acetamide
methyl 3-(2-methyl-1,3-thiazole-4-carbonyl)-7-oxo-9-[3-(pyridin-4-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(4-{[4-(4-hydroxy-2,8-dimethylquinolin-3-yl)butan-2-yl]amino}piperidin-1-yl)propan-1-one
1-[4-(furan-2-yl)pyrimidin-2-yl]-5-methyl-N,N-bis(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl (1R,5S,6R)-6-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}-3-azabicyclo[3.1.0]hexane-3-carboxylate
5-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-N,N,4-trimethylpyrimidin-2-amine
N-(1-{4-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)furan-3-carboxamide
5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)-1-(naphthalen-1-ylmethyl)pyrrolidin-2-one
2-(2,3-dihydro-1H-inden-1-yl)-N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}acetamide
2-(2,3-difluorophenoxymethyl)-N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-1,3-oxazole-4-carboxamide
methyl 3-[2-(1-ethyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]-4-methoxybenzoate
N-[2-(azepan-1-yl)ethyl]-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
2-{1-[4-(5-tert-butyl-1H-pyrazol-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}-3-methylpyridine
4-(1H-pyrazol-1-yl)-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
1-{[3-(cyclopentyloxy)phenyl]methyl}-3-(1-methyl-1H-imidazol-2-yl)piperidine
2-[1-cyclopentyl-3-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]acetamide
1-[(6-chloro-2-fluoro-3-methylphenyl)methyl]-3-methylimidazolidin-2-one
3-[2-(2-methoxyphenyl)pyrrolidin-1-yl]-N-(1,3-thiazol-2-yl)propanamide
3-[1-(methoxymethyl)cyclopentyl]-1-[3-(prop-2-en-1-yloxy)phenyl]urea
8-({2-[2-(dimethylamino)ethoxy]-3-methoxyphenyl}methyl)-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
N-{[7-(6-methoxypyridazin-3-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-methyl-1,2-oxazole-3-carboxamide