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3-(2H-1,3-benzodioxol-5-yl)-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]propanamide
2-methoxy-N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]benzamide
N-ethyl-N-[1-(4-methoxyphenyl)propyl]-3-(2-oxoimidazolidin-1-yl)benzamide
1-[(5-methylfuran-2-yl)methyl]-4-oxo-N3-(2-phenylethyl)-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[3-(pyridin-3-yloxy)propyl]acetamide
2-(2-chloro-4-{[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]methyl}phenoxy)acetamide
2-methyl-6-{2-[(2-methyl-1,3-thiazol-5-yl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
methyl (2S)-1-{2-[1-cyclopentyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetyl}pyrrolidine-2-carboxylate
1-(1'-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)propan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}furan-2-carboxamide
[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl){[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}amine
N-{[4-(3-methoxypiperidine-1-carbonyl)phenyl]methyl}-2-methylpropanamide
5-(2,5-difluorobenzenesulfonyl)-3-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
methyl 2-[(1-methylpiperidin-3-yl)methyl]-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
ethyl 1-{2-[1-benzyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetyl}piperidine-4-carboxylate
N-[4-(dimethylcarbamoyl)-2-methylphenyl]-3-(2-methoxyphenoxy)azetidine-1-carboxamide
N-[(2R,3R)-1'-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
N,3,4-trimethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-5-sulfamoylbenzamide
N-[3-(2,6-dimethylphenoxy)propyl]-N-methyl-1,2,5-oxadiazole-3-carboxamide
1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-N-{[4-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(2-hydroxyphenyl)acetamide
3-(4-{[4-(3,4-dimethylphenoxy)phenyl]methyl}piperazin-1-yl)propan-1-ol
2-[1-(4-chloro-2-methylphenyl)-5-[(2-oxopiperidin-1-yl)methyl]-1H-1,2,4-triazol-3-yl]acetamide
N-[3,3-dimethyl-1-(pyridin-3-yl)butyl]-6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(1,3-thiazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(4-fluorophenyl)-4-{4-[(3-oxopiperazin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}piperidine-1-carboxamide
methyl 2-{[1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidin-4-yl]formamido}-4-(methylsulfanyl)butanoate
3,5,7-trimethyl-2-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}-1H-indole
(1S,6R)-9-[1-(2-methoxyphenyl)piperidin-4-yl]-3,9-diazabicyclo[4.2.1]nonane
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(3-methylthiophen-2-yl)sulfonyl]piperidin-3-ol
8-methoxy-2-{[4-(pyridin-2-ylmethoxy)piperidin-1-yl]methyl}quinoline
2-(3-hydroxypiperidin-1-yl)-1-{4-[(2-methylphenyl)methyl]piperazin-1-yl}ethan-1-one
4-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}piperazine-1-carbaldehyde
5-[1-(4-methyl-2-oxopentanoyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
4-methoxy-N-(2-methoxyethyl)-2-{[1-(quinolin-8-ylmethyl)piperidin-4-yl]oxy}benzamide
(3S,4S)-1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[2-(pyridin-4-yl)acetyl]pyrrolidin-3-yl]acetamide
1-({4-methyl-5-[1-(1H-pyrrole-2-carbonyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
6-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
3-oxo-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-3,4-dihydroquinoxaline-2-carboxamide
1-benzyl-3-(2-methoxyethyl)-8-{[3-(2-methylphenyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[1-(furan-3-carbonyl)pyrrolidin-3-yl]-1-(2-phenylethyl)piperidine
3-{2-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-1-methyl-3-(4-phenylphenyl)pyrrolidine-2,5-dione
8-(1-methoxypropan-2-yl)-1-methyl-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[7-(3,6-dimethylpyrazin-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methoxybenzamide
2-(4-fluoro-2-methoxyphenyl)-2-{methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}acetic acid
N-cyclopropyl-1-[1-(2-phenylacetyl)piperidin-4-yl]piperidine-3-carboxamide
[2-({4-[(3,5-dichloropyridin-4-yl)methyl]piperazin-1-yl}methyl)phenyl]methanol
1-[4-(3-hydroxy-3-methylbutyl)benzoyl]-3-phenylpyrrolidin-3-ol