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N-[1-(7-{[5-(2-chlorophenyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-1-methylpiperidine-4-carboxamide
N-[2-(2-fluorophenoxy)phenyl]-4-methyl-3-oxo-2-(propan-2-yl)piperazine-1-carboxamide
(3aR,6aR)-2-(4-chloro-3-fluorobenzoyl)-5-(cyclobutylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-(pyridin-2-yl)pyrimidin-2-amine
2-(4-methoxyphenyl)-N-(thiophen-3-ylmethyl)acetamide
N-[(3R,5S)-1-cyclobutanecarbonyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-1-methyl-1H-pyrazole-5-carboxamide
4-(2,3-dihydro-1H-inden-2-yl)-11-[(pyridin-3-ylmethyl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-(1,2-oxazinan-2-yl)-N-[4-(oxolan-2-yl)butyl]propanamide
N-{7-[3-(diethylamino)pyrrolidine-1-carbonyl]-1-methyl-2-phenyl-1H-1,3-benzodiazol-5-yl}ethane-1-sulfonamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-5-(naphthalen-2-yl)-1,2,4-triazin-3-amine
2-[4-fluoro-2-(trifluoromethyl)phenyl]-6-(pyrrolidine-1-carbonyl)pyrazine
5-(8-methylquinolin-5-yl)pyrazin-2-amine
2-{[(4aS,8aS)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]methyl}-6,8-dimethyl-1,4-dihydroquinolin-4-one
8-({6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-2,8-diazaspiro[4.5]decan-3-one
6-(azepan-1-yl)-N-methyl-N-(oxan-4-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(pyridin-3-yloxy)ethyl]propanamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
4-{3-[(4S,4aS,8aR)-4-hydroxy-4-phenyl-decahydroquinoline-1-carbonyl]piperidin-1-yl}-2-(pyridin-4-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
3-[3-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2-methoxypyridine
7-(2-{[(3,5-dimethylphenyl)methyl]sulfanyl}acetyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
ethyl 1-{5-[(2-methylpropyl)carbamoyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carbonyl}piperidine-2-carboxylate
4-[(dimethyl-1,2-oxazol-4-yl)methyl]-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazine-2-carboxylic acid
6-{2-[(2-butyl-6-methylpyrimidin-4-yl)amino]ethyl}-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-[3-(benzyloxy)azetidin-1-yl]-2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)ethan-1-one
4-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]-2-methoxypyridine
3-(propoxymethyl)-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-1-carboxamide
2-[cyclopropyl(4-{3-methylimidazo[1,5-a]pyridin-1-yl}-1H-1,2,3-triazol-1-yl)methyl]-4-methylpyridine
2-methyl-N-{[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
ethyl 1-(2-phenylethyl)-5-(pyrazine-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
6-[(5-acetamidothiophen-2-yl)methyl]-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
5-[1-(cyclohexylmethyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
(2S,4S)-4-amino-1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-{2-[(3,5-dimethyladamantan-1-yl)oxy]ethyl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
2,3-dimethyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}quinoxaline-6-carboxamide
N-[2-(1H-indol-1-yl)ethyl]-2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}acetamide
1-(2-ethoxyethyl)-N,3-dimethyl-N-(quinolin-5-ylmethyl)-1H-pyrazole-5-carboxamide
{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine
N-(5-methyl-1,2-oxazol-3-yl)-2-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
1-cyclopentyl-N-[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
N-cyclopropyl-1-(1-{[(1-methyl-1H-pyrazol-4-yl)carbamoyl]methyl}piperidin-4-yl)piperidine-3-carboxamide
N-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}-1-propylpiperidin-4-amine
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
1-[(3-ethyl-1,2-oxazol-5-yl)methyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
5-ethyl-2-methyl-N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]pyrimidin-4-amine
N-cyclopropyl-3-(4-{[(2-methanesulfonamidoethyl)carbamoyl]amino}phenyl)propanamide
2-cyclopropyl-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
methyl 2-[2-(acetamidomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]benzoate
1-[(2-chlorophenyl)methyl]-N-methyl-N-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide