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N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N,5-dimethyl-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
2-(2-chloro-6-fluoro-3-methylphenyl)-1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-1H-imidazole
8-[(2,3-difluoro-6-methoxyphenyl)methyl]-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-({4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-4-(4-methylphenyl)benzamide
5-[(3-methoxyphenyl)methyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
2-methyl-N-[1-phenyl-2-(pyrrolidin-1-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
2-methyl-N-[3-(1,3-thiazol-4-yl)phenyl]-1,4-oxazepane-4-carboxamide
6-methyl-4-oxo-2-(2-phenylethyl)-1-(pyridin-2-ylmethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,4-dihydropyridine-3-carboxamide
N-(2,6-dimethylpyridin-3-yl)-4-[(3-methoxyphenyl)methyl]-3-oxopiperazine-1-carboxamide
3-[2-(3-acetylpiperidin-1-yl)-2-oxoethyl]-3-(2-fluorophenyl)-1-(2-methoxyethyl)pyrrolidine-2,5-dione
4-(1-{1-[2-(pyrrolidin-1-yl)benzoyl]piperidin-4-yl}ethyl)morpholine
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
5-chloro-4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-3-ethyl-1-methyl-1H-pyrazole
N-[(2-aminopyrimidin-5-yl)methyl]-N-methyl-6-(morpholin-4-yl)pyrimidin-4-amine
1-[(4-fluorophenyl)methyl]-4-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,4-diazepane
methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
7-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one
3-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
3-{5-[(3-hydroxy-4-methoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
2-methyl-5-{4-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
2-{4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}pyrazine
N-{2-[1-(1-cyclopentyl-6-oxopiperidine-3-carbonyl)piperidin-4-yl]ethyl}acetamide
N-[2-(2,3-dimethoxyphenyl)ethyl]-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
5-{[4-cyclohexyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-2-methoxyphenol
methyl (2S,4R)-1-[(2,4-difluorophenyl)methyl]-4-(quinoline-2-amido)pyrrolidine-2-carboxylate
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
1-{2-[(3-chlorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methyl-N-(1-methylpiperidin-4-yl)piperidine-4-carboxamide
4-[1-(2-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]pyridin-1-ium-1-olate
[(3R,4R)-1-[4-methyl-2-(pyridin-3-yl)pyrimidine-5-carbonyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
5-[1-(2-oxo-2-phenylacetyl)piperidin-4-yl]-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
(8aS)-2-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
(2E)-3-(3-fluorophenyl)-1-[4-(3-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]prop-2-en-1-one
1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N,N-dimethylazepan-4-amine
{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
(2S,4R)-1-[(2-aminopyridin-3-yl)methyl]-N,N-diethyl-4-[2-(methylsulfanyl)acetamido]pyrrolidine-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-{[(6-methylpyridin-2-yl)methyl]amino}piperidin-1-yl)benzamide
2-cyclopropyl-5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyrimidine
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-amino-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-5,6,7,8-tetrahydroquinazoline-4-carboxamide
1-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methylphenyl)-1,4-diazepane
2-methoxy-4-[1-(3-methylbutyl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
N-cycloheptyl-5-methyl-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-amine
1-[(1R,5S,8R)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]-2-(2-methoxyphenyl)ethan-1-one
(4aS,7aR)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-methyl-2-(morpholin-4-yl)propyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N,1-dimethyl-N-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-amine
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[4-(2-methoxyphenyl)-1,3-dimethyl-1H-pyrazol-5-yl]-1-methylurea
{1-[(5-chlorothiophen-2-yl)methyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
4-(3-benzyl-1H-pyrazol-5-yl)-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidine
1-[(3-chlorophenyl)methyl]-4-(3,3,3-trifluoro-2-methylpropyl)piperazine