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N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanamide
3-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propanamide
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methylpyrimidine-5-carboxamide
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(furan-2-carbonyl)piperazine
2-[(pyridin-4-ylmethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-[(2-fluorophenyl)methyl]-2-methyl-3-[2-(morpholin-4-yl)-2-oxoethyl]-4,5,6,7-tetrahydro-1H-indol-4-one
1-cyclopentyl-4-[4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one
methyl 3-[(4-methylphenyl)methyl]-7-oxo-9-(thiophen-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
[(2-fluorophenyl)methyl]({[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl})amine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyloxane-2-carboxamide
2-cyclopropanecarbonyl-8-(2-hydroxy-5-methylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{[5-methyl-2-(2-phenylmethanesulfonamidophenyl)-1,3-oxazol-4-yl]methyl}-2-(1,3-thiazol-4-yl)acetamide
methyl 6-[({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}carbamoyl)amino]-1,2,3,4-tetrahydroquinoline-1-carboxylate
N-(3-methoxyphenyl)-5-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
N-propyl-N-(pyridin-4-ylmethyl)-2,3-dihydro-1,4-benzodioxine-2-carboxamide
1-[2-(pyridin-4-yl)acetyl]-4-(1H-1,2,3-triazol-4-ylmethyl)-1,4-diazepane-6-carboxylic acid
1-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-[4-(propan-2-yl)morpholin-2-yl]ethan-1-one
3-(2-hydroxyphenyl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1H-pyrazole-5-carboxamide
(3aS,6aS)-2-cyclopentanecarbonyl-5-[5-(propan-2-yl)pyrimidin-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{[ethyl({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl})amino]methyl}-8-fluoroquinolin-4-ol
1-(benzyloxy)-8-(3,3-dimethylbutanoyl)-1,8-diazaspiro[4.5]decan-2-one
methyl[(3-methylphenyl)methyl]{[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-5-methyl-1,2-oxazole-3-carboxamide
2-{[4-(dimethylcarbamoyl)-6-hydroxy-1,4-diazepan-1-yl]methyl}benzoic acid
(2R,6S)-2,6-dimethyl-4-[4-(4-methylphenyl)-5-(pyrimidin-5-yl)pyrimidin-2-yl]morpholine
6-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]-4-tert-butyl-1,2-dihydropyrimidin-2-one
N-(3,3-diphenylpropyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
5-ethyl-2-{[3-(pyridine-2-carbonyl)piperidin-1-yl]methyl}pyridine
4-(5-fluoro-1H-indole-2-carbonyl)-1-(oxan-4-ylmethyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
1-{2-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]phenyl}ethan-1-one
1-cyclopropyl-3-[2-(2-ethylpiperidin-1-yl)-2-oxoethyl]-3-(2-methylphenyl)pyrrolidine-2,5-dione
1-(3,5-dimethylphenyl)-4-[(1-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-one
2-[3-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)phenyl]-3H,4H,5H,6H,7H,8H,9H-cyclohepta[d]pyrimidin-4-one
1-[(4-chlorophenyl)methyl]-N-[1-(methoxymethyl)cyclopentyl]-6-oxopiperidine-3-carboxamide
3-[3-({[1-(4-hydroxyphenyl)-2-methylpropan-2-yl]carbamoyl}amino)phenyl]-N-methylpropanamide
N-{3-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}-2-(naphthalen-2-yl)acetamide
3-(4-chlorophenyl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-3-phenylpropanamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-3,5-difluoro-N-methylbenzamide
5-{3-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridin-1-yl]-3-oxopropyl}imidazolidine-2,4-dione
8-(3-carboxy-4,6-dimethylpyridin-2-yl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[(2R,3R)-1'-[(2E)-3-(2,3-difluorophenyl)prop-2-enoyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N-cyclopropyl-1-ethyl-5-methyl-N-(3-phenylprop-2-yn-1-yl)-1H-pyrazole-4-carboxamide
N-methyl-2-(2-oxoazepan-1-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
1-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}-2-(pyridin-3-yl)ethane-1,2-dione
6-ethyl-1-methyl-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{[4-(naphthalen-1-yl)-4H-1,2,4-triazol-3-yl]methyl}phenol
(4aS,7aR)-1-[2-(methylamino)acetyl]-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-{1-[(2,5-dimethylphenyl)methyl]-4-hydroxypiperidin-4-yl}-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
N-[2-(2,4-difluorophenyl)-1-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]ethyl]-N-methylpyridine-3-carboxamide
2-(2,5-dimethylphenyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide