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2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]acetamide
N-(4-fluoro-2-methylphenyl)-3-{1-[(3-methyl-1H-indol-2-yl)methyl]piperidin-3-yl}propanamide
7-(2-hydroxyethyl)-2-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-ethyl-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyrrolidin-1-yl)ethyl]acetamide
1-methyl-N-({5-methyl-2-[3-(3-methylbutanamido)phenyl]-1,3-oxazol-4-yl}methyl)cyclopropane-1-carboxamide
4-cyclobutyl-6-methyl-N-[2-(pyrrolidin-1-yl)ethyl]pyrimidin-2-amine
N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-1,9-dioxaspiro[5.5]undecan-4-amine
(2R)-N-{4-[ethyl(phenyl)carbamoyl]phenyl}-2-(methoxymethyl)pyrrolidine-1-carboxamide
5-[3-(trifluoromethoxy)phenyl]pyridine-3-carboxamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(2,4-diethoxy-3-methylphenyl)methyl]-4-(hydroxymethyl)azepan-4-ol
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(piperidin-1-yl)ethyl]acetamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(pyridin-4-ylmethyl)acetamide
2-{4-[(2,4-dimethylphenyl)methyl]-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
5-{[1-(4-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-2-methyl-1,3-thiazole
2-(ethoxymethyl)-N,7-dimethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)[(3-methylpyridin-4-yl)methyl]amine
4-(4-{[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)amino}piperidin-1-yl)-N-[(2-fluorophenyl)methyl]benzamide
[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]({[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl})amine
N-{[3-methyl-7-(2-methylbenzoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-3-carboxamide
3-methyl-1-(2-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}-2-oxoethyl)-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(1R)-1-(3-methoxyphenyl)ethyl]propanamide
7-(2,3-dihydro-1,4-benzodioxin-6-yl)-1,2,3,4-tetrahydroisoquinoline
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-(2-methylpropyl)-1,2-oxazole-3-carboxamide
2-(4-chlorophenyl)-4-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}morpholine
3-(2,3-dihydro-1H-inden-2-yl)-5-methyl-5-{1-[2-(1,3-thiazol-4-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
2-[1-benzyl-4-(cyclohexylmethyl)piperazin-2-yl]ethan-1-ol
N-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-phenylbenzamide
N-{2-[(4-chlorophenyl)methoxy]ethyl}-2,2-dimethylcyclopropane-1-carboxamide
1-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-N-methylpiperidine-2-carboxamide
7-(cyclobutylmethyl)-2-[2-(4-methyl-1,4-diazepan-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
(3aS,6aS)-2-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[1-(4-methoxyphenyl)propyl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-(1H-1,2,3-benzotriazole-5-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
2-[1-(2,2-dimethylpropyl)-4-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperazin-2-yl]ethan-1-ol
(4aR,8aR)-7-[(5-ethylpyridin-2-yl)methyl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
3-(3-methylthiophene-2-carbonyl)-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
N-[2-(1H-imidazol-1-yl)ethyl]-N-methyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
N-cyclopropyl-2-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}acetamide
1-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)-4-phenylpiperidine-4-carbonitrile
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1-[(4-fluorophenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
(3S,4R)-1-[(2-cyclohexylpyrimidin-5-yl)methyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)({2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl})amine
6-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}-2-methylpyrimidin-4-ol
N-({2-[3-(4-methoxybenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-5-methyl-1,2-oxazole-3-carboxamide
4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1-{thieno[3,2-d]pyrimidin-4-yl}piperidine
3-[1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)piperidin-3-yl]-1-(morpholin-4-yl)propan-1-one
N-[(3R,4S)-1-(cyclobutylmethyl)-4-cyclopropylpyrrolidin-3-yl]furan-3-carboxamide