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1-[3-({[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]-3-(4-ethylpiperazin-1-yl)propan-2-ol
8-(pyridin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-[(3,4-difluorophenyl)methyl]-3-(2-oxo-2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethyl)piperazin-2-one
1-[(2-chlorophenyl)methyl]-3-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-5-fluoroquinazolin-4-amine
1-(oxan-4-yl)-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
3-[(dimethylamino)methyl]-1-(1H-pyrrole-2-carbonyl)piperidin-3-ol
2-[3-(2-fluorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(oxolan-3-yl)acetamide
1-(3,5-dichloro-4-methylbenzoyl)-3-(3-methoxypropyl)piperidine
4-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-2-one
(4aS,7aR)-1-(3,5-dimethylbenzoyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{2-[5-(hydroxymethyl)-1,2,4-oxadiazol-3-yl]ethyl}-1-[4-methyl-3-(2-oxopyrrolidin-1-yl)phenyl]urea
methyl (2S,4R)-4-(4-phenylbenzamido)-1-(thiophen-2-ylmethyl)pyrrolidine-2-carboxylate
1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(pyridin-3-ylmethyl)piperazine
5-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine-2-carbonitrile
2-(2-aminoethyl)-N-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)quinazolin-4-amine
methyl 6-(2-{[3-(2-methoxyphenyl)propanamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)pyridine-3-carboxylate
N-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-5-propyl-1,3,4-oxadiazol-2-amine
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-N-(2-phenylethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
3-[3-(2-methoxyphenoxy)propyl]-3-methyl-1-[4-(methylsulfanyl)phenyl]urea
N-({8-[(2-fluorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-(2-methoxyphenoxy)acetamide
3-{5-[1-(4-methoxyphenyl)-1H-imidazol-2-yl]thiophen-3-yl}prop-2-yn-1-ol
(1-{2-[2-(4-methoxy-2,3-dimethylphenyl)-1H-imidazol-1-yl]ethyl}piperidin-2-yl)methanol
3-fluoro-N-{1-[1-(4-phenylbutanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
1-{4-[7-(1-hydroxy-2,2-diphenylethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]piperidin-1-yl}ethan-1-one
4-{[4-ethoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}piperazine-1-sulfonamide
1-[(3-methoxyphenyl)methyl]-5-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}piperidin-2-one
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
methyl 2-[(butan-2-yl)sulfamoyl]-6-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
(3S,7S,8aS)-7-{[(2,4-difluorophenyl)methyl]amino}-3-(hydroxymethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-methyl-5-{4-[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
N-[2-(1H-imidazol-1-yl)ethyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylacetamide
N-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
1-[(3-methoxyphenyl)methyl]-4-(morpholine-2-carbonyl)piperazin-2-one
2-{[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]methyl}quinoline
3-[5-(5-acetylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-1-[(2S,6S)-6-butyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]propan-1-one
2,2-dimethyl-N-{[5-methyl-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
methyl 3-[({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)carbamoyl]propanoate
4-[4-(2,4,6-trimethylphenyl)phenyl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(2S)-N-{[7-(1,3-benzothiazol-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-acetamidopropanamide
(1R,2R,6S,7S)-4-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]-4-azatricyclo[5.2.1.02,6]decane
1-[2-(1H-imidazol-1-yl)ethyl]-2-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazole
1-cyclopentyl-3-(3-fluorophenyl)-3-[2-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-oxoethyl]pyrrolidine-2,5-dione
6-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazine-1-carbonyl)-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
N-(3-cyano-4-methoxyphenyl)-4-(1,1-dioxo-1λ6-thiolan-3-yl)piperazine-1-carboxamide
9-methoxy-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-3-(1,2,5-thiadiazole-3-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl})amine
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-{2-methyl-1-[7-(4,4,4-trifluorobutanoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]propyl}pyridine-2-carboxamide