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2-phenyl-1-[7-(pyridin-3-yl)-9-[2-(thiophen-2-yl)ethoxy]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
6-fluoro-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-[4-(2-fluorophenoxy)phenyl]-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
N-methyl-6-(morpholin-4-yl)-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
2-(4-chloro-2-methylphenoxy)-N-{3-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]propyl}propanamide
1-(4-{3-[3-(trifluoromethyl)benzoyl]piperidine-1-carbonyl}thiophen-2-yl)ethan-1-one
1-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(thiophene-2-carbonyl)piperazine
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-8-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-{[3-methyl-7-(2,2,3,3-tetramethylcyclopropanecarbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-3-sulfonamide
2-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]pyridin-3-ol
methyl 2-oxo-1-(prop-2-en-1-yloxy)-8-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylate
1-methyl-3-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1,2-dihydroquinolin-2-one
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-3-phenoxypropanamide
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-[(2,3-dimethoxyphenyl)methyl]-1,2-oxazole-3-carboxamide
(2S,4R)-4-amino-1-[6-ethyl-2-(piperidin-1-yl)pyrimidin-4-yl]-N-methylpyrrolidine-2-carboxamide
5-methoxy-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N,1-dimethyl-1H-indole-2-carboxamide
2-(1,2-dimethyl-1H-imidazol-5-yl)-8-methoxy-3-(1H-pyrazol-1-ylmethyl)quinoline
N-[4-({[(2-methoxyphenyl)methyl]carbamoyl}methyl)phenyl]butanamide
1-(3-methyl-1,2-oxazole-5-carbonyl)-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-2-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-3-(4-methylphenyl)propanamide
1-(3-methoxyphenyl)-4-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperazin-2-one
4-{[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]methyl}-5-tert-butylfuran-2-carboxamide
1-{1-[(4-ethylphenyl)methyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl}cyclopropane-1-carboxamide
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-(2-chlorophenyl)-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylpropanamide
N-{[3-(4-fluorophenyl)oxolan-3-yl]methyl}-6-methylimidazo[2,1-b][1,3]thiazole-5-carboxamide
4-({1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-2-yl}methyl)morpholine
7-{1,3,6-trimethyl-1H-pyrazolo[3,4-b]pyridine-4-carbonyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
5-phenyl-4-{1-[4-(propan-2-yloxy)benzoyl]piperidin-4-yl}-2-(pyridin-3-yl)pyrimidine
N-[2-(dimethylamino)ethyl]-4-{[2-(3-methoxyphenyl)ethyl]amino}-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
(3aR,6aR)-2-methanesulfonyl-5-[(2E)-3-phenylprop-2-en-1-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(8-{[2-(trifluoromethyl)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]benzamide
(1S,5R)-N-[(4-chlorophenyl)methyl]-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[2-(3,4-dimethylpiperazin-1-yl)-2-oxoethyl]-3-(3-fluorophenyl)-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-{[4-(trifluoromethyl)phenyl]methyl}propanamide
5-[(4-fluorophenyl)methyl]-3-(oxolan-3-yl)-5-[1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidin-4-yl]imidazolidine-2,4-dione
(2E)-N-{[8-(3-methylbutanoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-3-(pyridin-2-yl)prop-2-enamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(5-methyl-1,2-oxazol-3-yl)methyl]piperidine-3-carboxamide
1-(3-methylbutyl)-3-(propan-2-yl)-8-{[4-(trifluoromethyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[1-(4-ethenylbenzoyl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
2-phenyl-5-(thiolan-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
ethyl 1-(oxan-4-yl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
1-[5-(2-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-(2-methylphenoxy)piperidine
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-3-(2,5-dioxoimidazolidin-4-yl)-N-methylpropanamide
5-ethyl-2,3-dimethyl-N-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
{4-methyl-5-[1-(1,3-thiazol-4-ylmethyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methanol
4-[(4-fluorophenyl)methyl]-1-(2-phenylacetyl)-3-(propan-2-yl)-1,4-diazepan-5-one