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2-hydroxy-1-{6-[(4-methylpiperazin-1-yl)sulfonyl]-1,2,3,4-tetrahydroisoquinolin-2-yl}propan-1-one
2-(2-methoxyphenyl)-1-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}ethan-1-one
1-[(3-methoxyphenyl)methyl]-N-methyl-N-(oxan-4-yl)-6-oxopiperidine-3-carboxamide
2-methyl-4-[2-(3-phenylpropyl)morpholine-4-carbonyl]-1H-1,3-benzodiazole
3-(2H-1,3-benzodioxol-5-yl)-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-phenylpropanamide
2-(6-methoxypyridin-3-yl)benzonitrile
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-methoxybenzamide
N-[4-(furan-2-yl)phenyl]-1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidine-3-carboxamide
ethyl 1-[(5-acetylthiophen-3-yl)methyl]-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
11-(cyclohexylamino)-4-(3-phenylpropyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[4-(pyrimidin-2-yloxy)piperidin-1-yl]ethan-1-one
7-(4-chlorophenyl)-2-(hydroxymethyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-(1,3-benzothiazol-2-yl)-1-[3-(4-methoxy-2-methylbenzoyl)piperidin-1-yl]propan-1-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-[2-(pyridin-2-yl)ethyl]propanamide
7-cyclopentyl-2-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2,7-diazaspiro[4.5]decan-6-one
1-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-[1-({[2-(furan-2-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]benzamide
N-[(3R,4R)-1-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]-3-hydroxypiperidin-4-yl]pyrazine-2-carboxamide
N-methyl-N-[(1S)-1-phenylethyl]-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
3-{2-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-[(3-methoxyphenyl)methyl]piperazin-2-one
N-{3-[2-(6-methylpyridin-2-yl)-1H-imidazol-1-yl]phenyl}pyridine-3-carboxamide
2-amino-4-[2-(benzylsulfanyl)pyrimidin-5-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
5-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-4-methyl-1,2,3-thiadiazole
1-(morpholin-4-yl)-2-{4-[4-(pyridin-3-yl)pyrimidin-2-yl]piperazin-1-yl}ethan-1-one
9-methoxy-4-(1-methylpiperidin-4-yl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]urea
4-ethoxy-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}pyrimidin-2-amine
1-[1-(3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
N-(1H-indol-4-ylmethyl)-5-methyl-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-amine
2-butyl-5-(morpholine-4-carbonyl)-1,3-benzoxazole
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[(3-fluorophenyl)methyl]pyrrolidin-3-yl]-1-methyl-1H-pyrazole-4-carboxamide
6-methyl-2-[(2-methylphenyl)methyl]-4-oxo-1-(pyridin-2-ylmethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1,4-dihydropyridine-3-carboxamide
N-[(2S)-1-hydroxy-3-phenylpropan-2-yl]-3,4-dimethyl-5-sulfamoylbenzamide
methyl 5-{[(2,5-dimethylphenyl)methyl]amino}-3-acetamido-1-ethyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-(1-{1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}piperidine-4-carbonyl)morpholine
2-(3-fluorophenyl)-N-(propan-2-yl)pyridine-4-carboxamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetamide
1-[6-(2-{[(furan-3-ylmethyl)(methyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)pyridin-3-yl]ethan-1-one
3-[3-(dimethylamino)propyl]-5-[1-(2-fluorobenzoyl)piperidin-4-yl]-5-[(2-methylphenyl)methyl]imidazolidine-2,4-dione
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-3-(morpholin-4-yl)benzamide
naphthalen-1-yl (7S,9aR)-7-ethyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
3-methyl-8-[3-(2-oxoazepan-1-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-[3-(hydroxymethyl)-8-methylquinolin-2-yl]thiophene-2-carboxylic acid
4-(4-{[2-(dimethylcarbamoyl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)benzamide
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl][(3-ethyl-1,2-oxazol-5-yl)methyl]methylamine
1-[9-methoxy-7-(6-methoxypyridazin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pent-4-en-1-one
[(2S,4R,5R)-5-(2-fluorophenyl)-1-methyl-4-[({2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)methyl]pyrrolidin-2-yl]methanol
(4aR,7aS)-1-benzyl-4-(2-methylfuran-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(5-{1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine