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N-[2-(2-methoxyacetyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-3-(2-methoxyphenyl)propanamide
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(1H-pyrazol-1-yl)acetamide
N-{3-[cyclopentyl(methyl)amino]propyl}-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
3-[(1-cyclobutylpiperidin-4-yl)oxy]-N-cyclopropyl-4-methoxybenzamide
(3R,4R)-1-(4-chloro-2-fluorobenzoyl)-3-cyclopropyl-4-methylpyrrolidin-3-ol
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(2-methyl-1,3-thiazol-4-yl)methyl]propanamide
N-[3-(4-fluorophenyl)phenyl]-1-(6-methylpyrimidin-4-yl)piperidine-3-carboxamide
4,5-dimethyl-6-[3-(piperidin-1-yl)azetidin-1-yl]pyrimidin-2-amine
(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-(1-methyl-1H-pyrrole-2-carbonyl)-8-azabicyclo[3.2.1]octane
2-[4-(hydroxymethyl)phenyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(4aR,7aS)-1-{2-[methyl(pyrazin-2-ylmethyl)amino]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(4-chloro-3-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}phenyl)acetamide
methyl 4-[5-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)-1,2,4-oxadiazol-3-yl]benzoate
3-{2-[(2-propyl-1,3-thiazol-4-yl)formamido]acetamido}propanoic acid
3-{4-[4-(pyrimidin-2-yloxy)phenyl]-1H-1,2,3-triazol-1-yl}propane-1,2-diol
2-methoxy-1-{1'-[2-(2-methylphenyl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
(3S,4S)-4-(4-methylpiperazin-1-yl)-1-[1-(pyridine-2-carbonyl)piperidin-4-yl]pyrrolidin-3-ol
2-(4-methyl-3-phenylpiperazine-1-carbonyl)-5-(1H-1,2,3,4-tetrazol-1-yl)phenol
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2-(1H-1,2,4-triazol-1-yl)acetamide
3-[(3R,4S)-3-amino-4-propylpyrrolidine-1-carbonyl]-5-methoxybenzoic acid
(3-benzyl-1-cyclopentanecarbonylpiperidin-3-yl)methanol
2-{[(4-cyclopentylpyrimidin-2-yl)amino]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
5-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}-3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazole
(3S,4S)-4-cyclopropyl-1-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)pyrrolidine-3-carboxylic acid
4-methyl-N-[1-(morpholine-4-carbonyl)piperidin-4-yl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
(1-{[4-chloro-2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-3-(2-phenylethyl)piperidin-3-yl)methanol
4-{2-methyl-6-[1-(4-methyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]pyrimidin-4-yl}morpholine
4-(pyrrolidine-1-sulfonyl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
{5-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]furan-2-yl}methanol
5-oxo-1-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]pyrrolidine-3-carboxylic acid
3-[(3R,4S)-4-(dimethylamino)-1-(2-methyl-5-sulfamoylbenzoyl)piperidin-3-yl]propanoic acid
N-[2-(cyclohex-1-en-1-yl)ethyl]-6-{[4-(pyrrolidin-1-yl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
N-[1-(4-fluorophenyl)ethyl]-4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
[(1-cyclopentylpiperidin-3-yl)methyl](1H-imidazol-2-ylmethyl)[2-(piperidin-1-yl)ethyl]amine
N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-{4-[(3,4-dimethoxyphenyl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
methyl 1-methoxy-2-oxo-8-[2-(3-phenyl-1H-1,2,4-triazol-5-yl)acetyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
2-[4-(2H-1,3-benzodioxol-5-yl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-N-methyl-N-[1-(thiophen-2-yl)ethyl]acetamide
N-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-N-methyl-1-(3-phenylpropyl)piperidin-3-amine
2-[4-(1-hydroxy-3-methylbutyl)piperidin-1-yl]-N-(propan-2-yl)pyridine-4-carboxamide
5-[1-(1H-imidazol-1-yl)ethyl]-3-(oxan-4-yl)-1-(2-phenylethyl)-1H-1,2,4-triazole
2-{4-[2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperazin-1-yl}acetamide
2-(4-methanesulfonylmorpholin-3-yl)-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
thiophen-2-yl(1-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidin-4-yl)methanol
N-{1-[7-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-3-phenylpropanamide
3-(1,3-benzothiazol-6-yl)-1-[(4-methanesulfonylmorpholin-2-yl)methyl]urea
1-[(6-chloropyridin-3-yl)methyl]-3-(2-ethoxyethyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
4-phenyl-5-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazole
1-(4-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)ethan-1-one
4-(1H-pyrazol-4-yl)-1-[4-(thian-4-yl)piperazin-1-yl]butan-1-one