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3-(4-benzylpiperazine-1-carbonyl)-2-ethyl-1-[(1-ethylpyrrolidin-2-yl)methyl]-6-methyl-1,4-dihydropyridin-4-one
2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-(thiophen-2-ylmethyl)benzamide
1-[2-(piperidin-1-ylmethyl)phenyl]-3-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}urea
1-{3-[4-({[2-(3-chlorophenyl)ethyl]amino}methyl)-2-methoxyphenoxy]-2-hydroxypropyl}piperidin-4-ol
(4aR,7aS)-1-(2-methoxyacetyl)-4-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(dimethylamino)-N-(3-methyl-1-{7-[2-(naphthalen-1-yl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)acetamide
2-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}benzoic acid
N-[2-(2-fluorophenyl)-1-{1-[3-(pyridin-3-yl)propanoyl]piperidin-4-yl}ethyl]-N-methylthiophene-3-carboxamide
3-[2-hydroxy-3-(2-methylphenoxy)propanoyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
1-{[2-({[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)phenyl]methyl}pyrrolidin-2-one
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({[3-(propan-2-yl)-4,5-dihydro-1,2-oxazol-5-yl]methyl})amine
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4,6-dimethylpyrimidin-2-yl)piperazin-2-one
1-(2-aminoethyl)-N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)-1H-1,2,3-triazole-4-carboxamide
(1-{[4-(2-cyclopropylquinoline-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidin-3-yl)methanol
methyl 3-{3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carbonyl}benzoate
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl][2-(2-fluorophenyl)-1-{1-[(4-methoxyphenyl)methyl]piperidin-4-yl}ethyl]methylamine
N,5-dimethyl-N-[2-(pyridin-2-yl)ethyl]-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N,N-dimethyl-2-{[2-(propylsulfanyl)acetamido]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-(3-fluoropyridin-2-yl)-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
4-[(2,4-dimethylphenyl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-methyl-8-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-phenyl-1-(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperidin-3-yl)ethan-1-one
1-(3-methylpyridin-4-yl)-4-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperazine
2-ethyl-4-(1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-phenyl-1H-imidazol-5-yl)pyrimidine
6-oxo-1-[2-(pyridin-2-yl)ethyl]-N-[2-(pyrrolidin-1-yl)ethyl]piperidine-3-carboxamide
2-[3-(2-chlorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]acetamide
4-(2-{2,7-diazaspiro[4.5]decan-7-yl}-2-oxoethyl)-5-methyl-2,3-dihydro-1H-pyrazol-3-one
methyl 2-(azepane-1-sulfonyl)-6-(3-phenylprop-2-ynoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(trifluoromethyl)phenyl]methyl}amine
N,N-dimethyl-2-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-3-carboxamide
6-{[(1s,4s)-4-aminocyclohexyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
5-acetyl-N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[(3,5-dimethoxyphenyl)methyl]-1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
2-{2-[4-(pyridin-3-yloxy)piperidin-1-yl]ethyl}-2H-indazole
4-(hydroxymethyl)-N-[3-(1H-imidazol-1-yl)propyl]-N-(pyridin-3-ylmethyl)benzamide
[(3-{[1-(4-methoxybenzenesulfonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(thiophen-2-ylmethyl)amine
7-(3-phenyl-1,2-oxazole-5-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
5-(4-acetyl-2-methoxyphenoxymethyl)-N,N-diethyl-1,2-oxazole-3-carboxamide
1-benzyl-4-[(3-methoxyphenyl)methyl]-1,4-diazepan-5-one
methyl 1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-4-carboxylate
2-(2-aminoethyl)-N-[2-(1-cyclopentylpiperidin-4-yl)ethyl]quinazolin-4-amine
(1R,5R)-6-propyl-N-[4-(trifluoromethoxy)phenyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-{1-[(3,4-difluorophenyl)methyl]piperidin-3-yl}-4-(4-methoxyphenyl)piperazine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(6-ethoxy-4-methylquinazolin-2-yl)-N-methylpyrrolidine-2-carboxamide
1-(4-fluoro-2-methylbenzoyl)-3-(2-methoxyphenoxy)azetidine
N-(1-cycloheptylpiperidin-3-yl)-2-(1H-indazol-1-yl)acetamide
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(oxolan-2-ylmethyl)-N-propylbutanamide
4-(1-{1-[(4-chloro-3-fluorophenyl)methyl]piperidin-4-yl}ethyl)morpholine
1-{3-[5-(2-chlorophenyl)pyrimidin-4-yl]piperidin-1-yl}-2-(3,4,5-trimethoxyphenyl)ethan-1-one