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(4aS,8aR)-2-{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-decahydroisoquinoline
3-(3-fluorophenyl)-N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide
4-(4-methyl-1H-pyrazol-1-yl)-1-(pyrrolidine-1-carbonyl)piperidine-4-carboxylic acid
2-(pyridin-3-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}-2-(pyrrolidin-1-yl)acetamide
methyl 3-{[(1,3-dimethyl-1H-pyrazol-5-yl)formamido]methyl}-5-propanamidobenzoate
3-[ethyl({[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl})amino]-1λ6-thiolane-1,1-dione
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2,2,3-trimethylbut-3-enamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-[2-(6-methylpyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
3-{[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]methyl}benzonitrile
N-methyl-4-{[({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]methyl}benzamide
5-{2-[4-(2,3-dichlorophenyl)-1H-1,2,3-triazol-1-yl]ethyl}-1,3,4-thiadiazol-2-amine
(1S,5R)-6-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[1-(6-methyl-1,3-benzothiazol-2-yl)piperidin-4-yl]piperidin-3-ol
4-(piperidin-1-yl)-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]benzamide
2-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)acetamide
6-[2-(2,3-difluoro-6-methoxyphenyl)-1H-imidazol-1-yl]-3-ethyl-2,3-dihydro-1,3-benzoxazol-2-one
N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
3-(naphthalene-1-carbonyl)-1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperidine
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-3-yl]propan-1-ol
(1S,5R)-3-(2-amino-6-ethyl-5-methylpyrimidin-4-yl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 7-oxo-9-(3-phenylpropoxy)-3-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(1-methyl-1H-pyrazol-4-yl)methyl](propan-2-yl)amine
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-4-(3-methoxypropyl)piperazine
4-(2-methylphenoxy)-1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(1-methyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
methyl 7-oxo-3-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-chloro-4-[5-(dimethylamino)-1H-1,2,4-triazol-3-yl]benzamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-1H-indazole-3-carboxamide
1-[4-({[3-(4-fluorophenyl)oxolan-3-yl]methyl}amino)phenyl]-3-methylimidazolidin-2-one
3-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-1-[2-(propylsulfanyl)phenyl]urea
N-(1,4-dioxan-2-ylmethyl)-1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-amine
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propanamide
1-(3,4-dimethoxybenzoyl)-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
1-(2-methoxyethyl)-3-(2-methoxyphenyl)-3-{2-[4-(4-methoxyphenyl)piperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
1-methyl-3-phenyl-8-(piperidin-4-yl)-1,8-diazaspiro[4.5]decane
5-[1-(2-chlorobenzoyl)piperidin-4-yl]-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
4-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
4-{[2-(cyclohex-1-en-1-yl)ethyl]amino}-N-(2-hydroxyethyl)pyridine-2-carboxamide
3-phenoxy-N-{1-[1-(4,4,4-trifluorobutanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
methyl 2-(4-{1-[N-methyl-1-(1-methyl-1H-pyrazol-3-yl)formamido]-2-phenylethyl}piperidine-1-carbonyl)benzoate
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}[2-(4-methyl-1H-imidazol-2-yl)ethyl]amine
4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}-N,N-dimethylpiperidine-1-sulfonamide
4-methoxy-N-{[7-(methylsulfanyl)-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
1-(cyclopropylmethyl)-4-[5-(methoxymethyl)furan-2-carbonyl]-2-(propan-2-yl)-1,4-diazepane
3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-[2-(oxan-2-yl)ethyl]propanamide
N-[1-(4-chlorophenyl)-3-hydroxypropan-2-yl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
N-[2-(4-fluorophenyl)ethyl]-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2,5-difluoro-N-[1-(7-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]benzamide