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(1S,5R)-N-(2,5-dimethylphenyl)-6-(3-methylbut-2-en-1-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
6-(benzyloxy)-1-(2-methylpropyl)-4-(1,3-thiazole-5-carbonyl)-1,4-diazepan-2-one
2-(2-chloro-6-fluorobenzamido)-N-cyclohexyl-N-methyl-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
ethyl 4-[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]piperazine-1-carboxylate
3-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-1-methyl-1,2,5,6,7,8-hexahydroquinolin-2-one
methyl 3-{[2-(2-chlorophenyl)acetamido]methyl}-5-(furan-2-amido)benzoate
2-methoxy-N-(1-{7-[(4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
[3-(3-phenylpropyl)-1-[6-(propan-2-yl)pyrimidin-4-yl]piperidin-3-yl]methanol
N-(2-methyl-1-{7-[(2-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)furan-3-carboxamide
N-[(3R,4R)-3-hydroxy-1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidin-4-yl]pyrazine-2-carboxamide
4-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,2-dihydroquinazolin-2-one
4-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidin-2-amine
N-(furan-2-ylmethyl)-N-methyl-3-(2-methyl-1H-indol-1-yl)propanamide
N4,N4,N6-trimethyl-N6-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrimidine-4,6-diamine
3-[4-methyl-2-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenyl]-1,3-oxazolidin-2-one
7-(3-chlorophenyl)-4-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
2-(3-chlorothiophene-2-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
methyl(2-phenyl-1-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}ethyl)(pyridin-3-ylmethyl)amine
(3R,9aR)-8-[(4-methoxyphenyl)methyl]-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{2-methyl-5-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]phenyl}imidazolidin-2-one
6-[(3,3-diethylpyrrolidin-1-yl)methyl]-N-(1,4-dioxan-2-ylmethyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
N-ethyl-4-oxo-2-phenyl-1,3,8-triazaspiro[4.5]dec-1-ene-8-carboxamide
methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl][(2,3,4-trifluorophenyl)methyl]amine
2-{1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}-1H-1,3-benzodiazole
8-[(3,5-dichloropyridin-4-yl)methyl]-2-(dimethylamino)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
(2R,3R,6R)-3-(4-fluorophenyl)-5-(1-methyl-1H-indazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-cyclohexyl-N3-cyclopropyl-N5-[(2,4-dimethoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-(3-{[6-(piperidin-1-yl)pyrimidin-4-yl]amino}propyl)pyrrolidine-2,5-dione
N-[5-(3-methylpiperidine-1-carbonyl)-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazol-7-yl]acetamide
2,4-dimethyl-N-{[7-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,3-thiazole-5-carboxamide
N-[(2R,3R)-2-methoxy-1'-{[4-(methylsulfanyl)phenyl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
1-(isoquinolin-5-yl)-3-{[1-(morpholin-4-yl)cyclopentyl]methyl}urea
3-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-[(2-fluorophenyl)methyl]propanamide
2-[(cyclopropylmethyl)sulfanyl]-1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
N-[cyclopropyl(1-methyl-1H-1,2,4-triazol-5-yl)methyl]-6-ethylpyrimidin-4-amine
N-[2-methyl-5-({[2-(2-oxopiperidin-1-yl)ethyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
methyl({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
8-(4-methyl-1,3-thiazole-5-carbonyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
2-(3-methylbutyl)-8-[2-(morpholin-4-yl)-2-oxoethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-amino-N-cyclopropyl-3-ethyl-N-[(3-hydroxyphenyl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(5-methylpyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(3R,4S)-1-(5-chloropyridin-2-yl)-4-propylpyrrolidin-3-amine
6-(3-fluoro-4-methoxybenzoyl)-N-(2-methyl-1,3-benzothiazol-5-yl)-6-azaspiro[2.5]octane-1-carboxamide
methyl 3-({[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]carbamoyl}amino)-4-methoxybenzoate
3-(3,4-dimethoxyphenyl)-1-{4-[2-(pyridin-2-yl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}propan-1-one
1-methyl-3-(propan-2-yl)-5-[2-(trifluoromethyl)pyrrolidine-1-carbonyl]-1H-pyrazole
N4-methyl-6-(morpholin-4-yl)-N4-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)pyrimidine-2,4-diamine
N-methyl-2-(2-phenylethyl)-N-(pyridin-3-ylmethyl)-1,3-benzoxazole-5-carboxamide
N,N-dimethyl-2-(4-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-1,4-diazepan-1-yl)acetamide