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ethyl 2-(1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)acetate
N-({8-[(2-fluorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)oxolane-2-carboxamide
(3aS,6aR)-3-[2-(4-methoxyphenyl)ethyl]-5-(1,3-thiazol-2-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-(cyclohexylmethyl)-6,7-dimethoxy-3-({[(trimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
5-acetyl-N-{[3-methyl-7-(1H-pyrazole-4-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-3-carboxamide
N-[4-(3-fluorophenyl)phenyl]-1-(2-methylfuran-3-carbonyl)piperidine-3-carboxamide
(5S,9aS,9bS)-2-cyclopentyl-5-(3-methyl-1H-indol-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-N-[3-(1H-indol-2-yl)phenyl]piperidine-3-carboxamide
2-{[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1-propyl-1H-imidazole
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-imidazole-2-carbonyl)piperidine
1-{3-[(2-methoxyphenyl)methyl]-5-(propan-2-yl)-1H-1,2,4-triazol-1-yl}butan-2-ol
dimethyl({1-[3-(quinolin-6-yl)phenyl]ethyl})amine
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
(2S)-2-[2-(3-hydroxyadamantan-1-yl)acetamido]-3-(4-hydroxyphenyl)propanamide
3-(2,3-dihydro-1-benzofuran-7-yl)-6-(propan-2-yloxy)pyridazine
1-(cyclopropylmethyl)-N-methyl-5-[2-(1-methyl-1H-pyrrol-3-yl)acetyl]-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-(4-benzylpiperazine-1-carbonyl)-1-(butan-2-yl)-N-(furan-2-ylmethyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-(2-phenylethyl)-4-[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperazin-2-one
2-(1-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-imidazol-2-yl)-4,5,6,7-tetrahydro-1,3-benzothiazole
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)propanamide
2-[(4aR,7aS)-4-[(cyclohexylmethyl)carbamoyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
6-[3-hydroxy-3-(piperidin-1-ylmethyl)pyrrolidin-1-yl]pyridine-3-carbonitrile
N-(oxolan-2-ylmethyl)-3-{1-[2-(phenylsulfanyl)acetyl]piperidin-4-yl}propanamide
(3S,4S)-1-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-4-propylpyrrolidine-3-carboxylic acid
8-[(3-hydroxyphenyl)methyl]-1-(3-methylbutyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(2-chlorophenyl)methyl]-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-(4-fluorophenyl)-1-[1-(propan-2-yl)piperidine-4-carbonyl]piperidin-3-amine
N-[2-(methylsulfanyl)ethyl]-1-[2-(morpholin-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
6-(methylsulfanyl)-2-(piperidin-3-ylmethyl)-1,2,3,4-tetrahydroisoquinoline
(3aS,6aR)-N,N-dimethyl-2-oxo-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-sulfonamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-methyl-N-[2-(4-methylphenoxy)ethyl]benzamide
4-hydroxy-4-(1H-imidazol-1-ylmethyl)-N-(5,6,7,8-tetrahydronaphthalen-1-yl)piperidine-1-carboxamide
1-(cyclohexylmethyl)-4-[(quinoxalin-2-yl)amino]pyrrolidin-2-one
(1H-imidazol-2-ylmethyl)(methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
3-[2-(dimethylamino)ethyl]-8-[(1-methyl-1H-indol-3-yl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{2-[4-(2,5-dimethoxyphenyl)-4H-1,2,4-triazol-3-yl]ethyl}phenol
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,3-oxazole-4-carboxamide
(3S,9aR)-3-benzyl-8-(4-chlorobenzoyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(5-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
1-[5-({[(3,5-difluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
3-chloro-N-cyclopentyl-N-({3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)benzamide
(2S)-1-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-{3-[5-(2-fluorophenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}-4-methylpentan-1-one
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-3-(pyrazin-2-yl)propan-1-one
2-(dimethyl-1,3-thiazol-5-yl)-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]acetamide
(1R,5R)-N,N-dimethyl-6-[(1-methyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
(3R,4R)-1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-ol
1-(cyclohexylmethyl)-N-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}piperidin-3-amine